SCHEMBL8326465

SCHEMBL8326465

CN1CCc2c(ccc3c2NC(=O)C3=O)C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 3/20 0.40
MAOA P21397 2/20 0.39
MAOB P27338 2/20 0.39
DAO P14920 2/20 0.38
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
PRKCB P05771 2/20 0.35
GSK3B P49841 2/20 0.35
PRKCG P05129 1/20 0.35
PRKCA P17252 1/20 0.35
PRKCE Q02156 1/20 0.35
PRKCD Q05655 1/20 0.35
BRD4 O60885 1/20 0.35
BRD9 Q9H8M2 1/20 0.35
NSD2 O96028 1/20 0.35
BCHE P06276 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
DRD1 P21728 1/20 0.35
DRD5 P21918 1/20 0.35
CRBN Q96SW2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327753 0.86 CES1 (0.42) CES1DAONSD2BCHEL3MBTL1
SCHEMBL8325695 0.82 MAOA (0.34) MAOAMAOBHSP90AA1HSP90AB1PRKCB
SCHEMBL8325697 0.82 MAOA (0.34) MAOAMAOBHSP90AA1HSP90AB1PRKCB
SCHEMBL8328296 0.81 NOTUM (0.46) CES1GSK3B
SCHEMBL8325983 0.75 ESR1 (0.48) CES1
SCHEMBL2254584 0.74 PARP1 (0.53) CES1DAONSD2BCHE
SCHEMBL2251074 0.74 PARP1 (0.57) CES1MAOAMAOBDAONSD2
SCHEMBL4350619 0.74 ALDH1A1 (0.44) CES1BCHE
SCHEMBL13232796 0.74 CES1 (0.36) CES1L3MBTL1
SCHEMBL8331316 0.73 CES1 (0.40) CES1DAONSD2BCHEL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529636-B1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH AS (DK) 1999-06-23 EP disclosed
US-5436250-A Isatineoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1995-07-25 US disclosed
US-5242918-A Isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-09-07 US disclosed
WO-1993005043-A1 NOVEL ISATINOXIME DERIVATIVES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 1993-03-18 WO disclosed
EP-0529636-A1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-03-03 EP disclosed