SCHEMBL8328296

SCHEMBL8328296

CC(=O)N1CCc2c(ccc3c2NC(=O)C3=O)C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.46
HRH3 Q9Y5N1 1/20 0.39
BAZ2B Q9UIF8 5/20 0.38
MAPT P10636 2/20 0.38
LMNA P02545 1/20 0.38
LCK P06239 5/20 0.37
RET P07949 5/20 0.37
KDR P35968 5/20 0.37
LRRK2 Q5S007 4/20 0.37
ALK Q9UM73 4/20 0.37
PDGFRA P16234 4/20 0.37
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37
ALDH1A1 P00352 1/20 0.36
ALOX15 P16050 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CES1 P23141 1/20 0.36
EP300 Q09472 1/20 0.36
CREBBP Q92793 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2257179 0.90 NOTUM (0.46) NOTUMHRH3BAZ2BMAPTLMNA
SCHEMBL8325734 0.85 NOTUM (0.42) NOTUMHRH3BAZ2BMAPTLMNA
SCHEMBL8325730 0.85 NOTUM (0.42) NOTUMHRH3BAZ2BMAPTLMNA
SCHEMBL8325983 0.84 ESR1 (0.48) CES1EP300CREBBPLIG1
SCHEMBL8326465 0.81 CES1 (0.40) GSK3BCES1
SCHEMBL8329492 0.73 BAZ2B (0.43) BAZ2BMAPTLCKRETKDR
SCHEMBL2255155 0.73 NOTUM (0.50) NOTUMMAPTALDH1A1CES1LIG1
SCHEMBL8327753 0.73 CES1 (0.42) ALDH1A1CES1LIG1
SCHEMBL2254584 0.70 PARP1 (0.53) CES1LIG1
SCHEMBL2251074 0.70 PARP1 (0.57) CES1LIG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529636-B1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH AS (DK) 1999-06-23 EP disclosed
US-5436250-A Isatineoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1995-07-25 US disclosed
US-5242918-A Isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-09-07 US disclosed
WO-1993005043-A1 NOVEL ISATINOXIME DERIVATIVES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 1993-03-18 WO disclosed
EP-0529636-A1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-03-03 EP disclosed