SCHEMBL8330144

SCHEMBL8330144

CCOC(=O)CN1CCc2c(ccc3c2NC(=O)C3=NO)C1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 2/20 0.37
PDCD1 Q15116 1/20 0.37
PIN1 Q13526 1/20 0.36
PIN4 Q9Y237 1/20 0.36
LMNA P02545 3/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
HSD17B10 Q99714 1/20 0.34
AOC3 Q16853 2/20 0.33
ALOX15 P16050 1/20 0.32
CA12 O43570 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
MEN1 O00255 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8330143 1.00 CD274 (0.37) CD274PDCD1PIN1PIN4LMNA
SCHEMBL8327099 0.88 CD274 (0.39) CD274PDCD1PIN1PIN4LMNA
SCHEMBL8331250 0.77 PNMT (0.30)
SCHEMBL8325695 0.77 MAOA (0.34) LMNASMN1; SMN2ALDH1A1KDM4EMAPT
SCHEMBL8331247 0.77 PNMT (0.30)
SCHEMBL8325697 0.77 MAOA (0.34) LMNASMN1; SMN2ALDH1A1KDM4EMAPT
SCHEMBL8325730 0.76 NOTUM (0.42) LMNAMAPTGSK3AGSK3B
SCHEMBL8325734 0.76 NOTUM (0.42) LMNAMAPTGSK3AGSK3B
SCHEMBL8329197 0.72 ESR1 (0.44)
SCHEMBL3841321 0.71 HDAC1 (0.37) CD274PDCD1LMNASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529636-B1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH AS (DK) 1999-06-23 EP disclosed
US-5436250-A Isatineoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1995-07-25 US disclosed
US-5242918-A Isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-09-07 US disclosed
WO-1993005043-A1 NOVEL ISATINOXIME DERIVATIVES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 1993-03-18 WO disclosed
EP-0529636-A1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-03-03 EP disclosed