SCHEMBL8327245

SCHEMBL8327245

Cc1ccc(S(=O)(=O)n2cnc3ccccc32)c(C)c1

nearest known ligand 0.80

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.80
TSHR P16473 3/20 0.80
KMT2A Q03164 3/20 0.68
NPC1 O15118 1/20 0.66
POLB P06746 4/20 0.66
ALDH3A1 P30838 4/20 0.66
NOD1 Q9Y239 1/20 0.66
L3MBTL1 Q9Y468 1/20 0.66
SMN1; SMN2 Q16637 3/20 0.65
GAA P10253 3/20 0.56
MEN1 O00255 2/20 0.56
PKM P14618 1/20 0.56
ALDH1A1 P00352 2/20 0.54
TP53 P04637 1/20 0.54
USP2 O75604 1/20 0.52
LMNA P02545 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8330999 0.86 HTT (0.67) HTTTSHRKMT2ANPC1POLB
SCHEMBL17960655 0.83 HTT (0.69) HTTTSHRKMT2ANPC1POLB
SCHEMBL8329551 0.80 ALDH3A1 (1.00) HTTTSHRKMT2ANPC1POLB
SCHEMBL8324963 0.75 HTT (0.55) HTTTSHRKMT2ANPC1POLB
SCHEMBL3470648 0.75 ALOX5 (0.75) HTTTSHRKMT2ANPC1POLB
SCHEMBL19848205 0.74 HTT (0.69) HTTTSHRKMT2ANPC1POLB
SCHEMBL19911331 0.74 HTT (0.69) HTTTSHRKMT2ANPC1POLB
SCHEMBL422055 0.72 ALDH3A1 (0.77) HTTTSHRKMT2APOLBALDH3A1
SCHEMBL7100805 0.72 ALDH3A1 (0.61) HTTTSHRKMT2APOLBALDH3A1
SCHEMBL14919981 0.71 GAA (0.59) HTTTSHRKMT2ANPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869787-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-24 EP disclosed
EP-0869787-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-14 EP disclosed
WO-1997024119-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed