SCHEMBL8328159

SCHEMBL8328159

COc1c(C(=O)O)c2n(c1-c1cccnc1F)CCCC2O

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 4/20 0.37
FFAR4 Q5NUL3 4/20 0.33
SCN9A Q15858 1/20 0.33
PDE4A P27815 1/20 0.33
NAPRT Q6XQN6 1/20 0.33
IDO1 P14902 1/20 0.32
HCRTR1 O43613 2/20 0.32
HCRTR2 O43614 2/20 0.32
ABL1 P00519 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32
GSK3B P49841 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7964887 0.92 L3MBTL1 (0.33) DHODHFFAR4SCN9APDE4AHCRTR1
SCHEMBL7962621 0.91 ABL1 (0.35) SCN9APDE4AIDO1HCRTR1HCRTR2
SCHEMBL7963165 0.91 SCN9A (0.34) SCN9APDE4AHCRTR1HCRTR2ABL1
SCHEMBL8330824 0.89 DHODH (0.43) DHODHFFAR4NAPRTHCRTR1HCRTR2
SCHEMBL8328923 0.88 DHODH (0.37) DHODHIDO1HCRTR1HCRTR2KMT2A
SCHEMBL8330821 0.85 DHODH (0.36) DHODHFFAR4NAPRTABL1
SCHEMBL8327360 0.83 DHODH (0.35) DHODHFFAR4NAPRTHCRTR1ABL1
SCHEMBL7965300 0.82 KCNMA1 (0.34) PDE4AHCRTR1HCRTR2ABL1
SCHEMBL8327934 0.82 DHODH (0.35) DHODHFFAR4NAPRTABL1KMT2A
SCHEMBL7967665 0.82 ABL1 (0.35) DHODHIDO1HCRTR1HCRTR2ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946555-A1 PYRROLE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Aventis Pharma S.A. (FR) 1999-10-06 EP claimed
WO-1998025925-A1 PYRROLE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM RHONE-POULENC RORER S.A. (FR) 1998-06-18 WO claimed
EP-0946555-A1 PYRROLE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Aventis Pharma S.A. (FR) 1999-10-06 EP disclosed
WO-1998025925-A1 PYRROLE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM RHONE-POULENC RORER S.A. (FR) 1998-06-18 WO disclosed