SCHEMBL8328443

SCHEMBL8328443

CCOC(=O)CC1NC(=O)Cc2cc(OS(=O)(=O)C(F)(F)F)ccc21

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.42
DRD2 P14416 3/20 0.37
DRD3 P35462 3/20 0.37
HTR1D P28221 2/20 0.37
DRD1 P21728 2/20 0.36
DRD4 P21917 2/20 0.36
DRD5 P21918 2/20 0.36
HSD11B1 P28845 1/20 0.35
KMT2A Q03164 1/20 0.34
BRD4 O60885 2/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
ALDH1A1 P00352 2/20 0.33
ADORA1 P30542 1/20 0.33
HPGD P15428 1/20 0.33
HTR1A P08908 1/20 0.33
HTR1B P28222 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327308 0.82 KMT2A (0.45) CYP1A2DRD2DRD3HTR1DKMT2A
SCHEMBL9979558 0.77 PPARD (0.53) DRD2DRD3HTR1D
SCHEMBL4760401 0.75 PPARD (0.46) DRD2DRD3HTR1D
SCHEMBL5533444 0.72 DGAT1 (0.40) DRD2DRD3HTR1DDRD1DRD4
SCHEMBL2254801 0.72 DGAT1 (0.40) DRD2DRD3HTR1DDRD1DRD4
SCHEMBL14061800 0.72 CYP24A1 (0.48) DRD2DRD3HTR1D
SCHEMBL2254799 0.72 DGAT1 (0.40) DRD2DRD3HTR1DDRD1DRD4
SCHEMBL2253838 0.71 DGAT1 (0.39) DRD2DRD3HTR1DDRD1DRD4
SCHEMBL2253842 0.71 DGAT1 (0.39) DRD2DRD3HTR1DDRD1DRD4
SCHEMBL5536891 0.71 DGAT1 (0.39) DRD2DRD3HTR1DDRD1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869787-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-24 EP disclosed
EP-0869787-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-14 EP disclosed
WO-1997024119-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed