SCHEMBL8327308

SCHEMBL8327308

CCOC(=O)CC1NCCc2cc(OS(=O)(=O)C(F)(F)F)ccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.45
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40
CA9 Q16790 2/20 0.40
CA14 Q9ULX7 2/20 0.40
KDM1A O60341 4/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
DRD2 P14416 1/20 0.39
HTR1D P28221 1/20 0.39
DRD3 P35462 1/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
OPRM1 P35372 2/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
KDM6B O15054 2/20 0.38
KDM4C Q9H3R0 2/20 0.38
PPARD Q03181 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8469394 0.85 KMT2A (0.60) KMT2ACA1CA2CA7CA9
SCHEMBL8328443 0.82 CYP1A2 (0.42) KMT2ADRD2HTR1DDRD3CYP1A2
SCHEMBL9979558 0.82 PPARD (0.53) DRD2HTR1DDRD3PPARD
SCHEMBL8466120 0.80 KMT2A (0.47) KMT2ASMN1; SMN2MEN1MAPTHTT
SCHEMBL4760401 0.80 PPARD (0.46) DRD2HTR1DDRD3KDM4CPPARD
SCHEMBL8469298 0.80 KMT2A (0.48) KMT2ACA1CA2CA7CA9
SCHEMBL7334819 0.76 SMN1; SMN2 (0.57) KMT2ASMN1; SMN2MEN1MAPTHTT
Hydrochloric Acid SCHEMBL8470673 0.75 SMN1; SMN2 (0.56) KMT2ASMN1; SMN2MEN1MAPTHTT
SCHEMBL3382275 0.73 KMT2A (0.62) KMT2AKDM4C
SCHEMBL3383043 0.73 KMT2A (0.62) KMT2AKDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869787-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-24 EP disclosed
EP-0869787-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-14 EP disclosed
WO-1997024119-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed