SCHEMBL8328586

SCHEMBL8328586

CC(C[CH]c1cccc(Cl)c1)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
CHRM5 P08912 1/20 0.41
CYP1A2 P05177 2/20 0.39
CYP2C9 P11712 2/20 0.39
MEN1 O00255 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
TAAR1 Q96RJ0 2/20 0.39
MAOB P27338 1/20 0.39
IDO1 P14902 1/20 0.38
TDO2 P48775 1/20 0.38
CHAT P28329 1/20 0.38
GRIK1 P39086 1/20 0.38
GRIK2 Q13002 1/20 0.38
ADRB2 P07550 1/20 0.38
ADRB1 P08588 1/20 0.38
ADRB3 P13945 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326387 0.83 TAAR1 (0.41) ALDH1A1HPGDCYP3A4TAAR1
SCHEMBL14910878 0.82 TAAR1 (0.50) TAAR1
SCHEMBL8324571 0.82 TP53 (0.43) TAAR1ACP3RELA
SCHEMBL8324064 0.81 SCN4A (0.44) CHRM5MAOBIDO1TDO2GRIK1
SCHEMBL8322584 0.81 MAOA (0.49) TAAR1MAOBNPSR1
SCHEMBL8327482 0.80 CYP3A4 (0.42) ALDH1A1HPGDCYP1A2CYP2C9MEN1
SCHEMBL16950868 0.78 TSHR (0.45) CHRM5CYP1A2CYP2C9MAOBCHAT
SCHEMBL16957527 0.78 CHRM5 (0.47) CHRM5CYP1A2CYP2C9MEN1CYP2D6
SCHEMBL8324977 0.77 IDO1 (0.49) ALDH1A1CYP1A2CYP2C9MEN1CYP3A4
SCHEMBL1989041 0.73 CHRM5 (0.54) ALDH1A1CHRM5CYP1A2CYP2C9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed