SCHEMBL8324977

SCHEMBL8324977

CC(C[CH]c1cccc(C(F)(F)F)c1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.49
TDO2 P48775 2/20 0.49
NFE2L2 Q16236 1/20 0.44
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42
ACP3 P15309 2/20 0.41
PNMT P11086 1/20 0.41
ATM Q13315 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
POLB P06746 1/20 0.40
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8329048 0.83 NPC1 (0.46) HTR2AHTR2CHTR2BACP3MEN1
SCHEMBL8322926 0.82 IDO1 (0.52) IDO1TDO2NFE2L2HTR2AHTR2C
SCHEMBL8326387 0.80 TAAR1 (0.41) HTR2ASMN1; SMN2MAPTALDH1A1CYP3A4
SCHEMBL14910878 0.79 TAAR1 (0.50) HTR2A
SCHEMBL8324571 0.78 TP53 (0.43) ACP3SMN1; SMN2NPC1MAPTRAB9A
SCHEMBL8328586 0.77 ALDH1A1 (0.46) IDO1TDO2ACP3PNMTMEN1
SCHEMBL8322584 0.77 MAOA (0.49) HTR2ANPC1MAPTMAOB
SCHEMBL20821033 0.76 IDO1 (0.51) IDO1TDO2HTR2AHTR2CHTR2B
SCHEMBL6309987 0.76 NFE2L2 (0.56) NFE2L2HTR2AHTR2CHTR2BMEN1
SCHEMBL6703600 0.74 PNMT (0.47) IDO1TDO2HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed