SCHEMBL8328962

SCHEMBL8328962

COc1ccc(Cl)cc1CNN1CCCCC1c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 6/20 0.53
CFTR P13569 1/20 0.45
DRD2 P14416 3/20 0.41
DRD4 P21917 3/20 0.41
KMT2A Q03164 3/20 0.41
GAA P10253 1/20 0.41
CPT1A P50416 1/20 0.40
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 1/20 0.39
KDM1A O60341 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39
PSENEN Q9NZ42 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328961 1.00 TACR1 (0.53) TACR1CFTRDRD2DRD4KMT2A
SCHEMBL1626959 0.86 KMT2A (0.53) TACR1KMT2AGAAALDH1A1MEN1
SCHEMBL8611479 0.85 TACR1 (0.38) TACR1CFTRDRD2KMT2ACPT1A
Hydrochloric Acid SCHEMBL8613936 0.84 TACR1 (0.38) TACR1CFTRDRD2KMT2ACPT1A
SCHEMBL8681005 0.83 TACR1 (0.39) TACR1KMT2AGAAKDM1AMAOA
Hydrochloric Acid SCHEMBL8681079 0.82 TACR1 (0.39) TACR1KMT2AGAAKDM1AMAOA
Hydrochloric Acid SCHEMBL9420087 0.82 TACR1 (0.57) TACR1
SCHEMBL20178136 0.82 TACR1 (0.55) TACR1CFTRKDM1AMAOAMAOB
SCHEMBL20178205 0.81 TACR1 (0.46) TACR1CFTRKDM1AMAOAMAOB
SCHEMBL8701388 0.80 TACR1 (0.58) TACR1DRD2KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5990125-A NK-1 receptor antagonists for the treatment of cancer PFIZER INC. (US) 1999-11-23 US disclosed