SCHEMBL8329222

SCHEMBL8329222

CCCCc1cn(Cc2ccc(-c3ccccc3OC(=O)O)cc2)c2cc(C=O)ccc2c1=O

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ICMT O60725 4/20 0.42
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
P2RX3 P56373 1/20 0.38
AGTR1 P30556 3/20 0.38
AGTR2 P50052 2/20 0.38
CNR1 P21554 1/20 0.37
CHRM1 P11229 1/20 0.36
TOP1 P11387 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8324163 0.93 ICMT (0.45) ICMTTP53MAPTAGTR1AGTR2
SCHEMBL8327103 0.92 ESR1 (0.40) ICMTTP53MAPTP2RX3AGTR1
SCHEMBL8329353 0.91 ICMT (0.43) ICMTTP53MAPTP2RX3AGTR1
SCHEMBL8328934 0.89 CHRM1 (0.47) ICMTTP53CHRM1
SCHEMBL8325903 0.87 AGTR1 (0.52) AGTR1AGTR2
SCHEMBL8327081 0.85 ICMT (0.43) ICMTTP53MAPT
SCHEMBL8322474 0.84 AGTR1 (0.41) ICMTTP53MAPTAGTR1AGTR2
SCHEMBL8330654 0.84 ICMT (0.40) ICMTTP53MAPTAGTR1AGTR2
SCHEMBL8327393 0.81 AGTR1 (0.50) AGTR1AGTR2CHRM1
SCHEMBL8324160 0.80 AGTR1 (0.52) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0498721-B1 N-substituted quinoline derivatives, process for their preparation, their use as pharmaceuticals and pharmaceutical compositions containing them HOECHST MARION ROUSSEL INC (FR) 1999-12-22 EP claimed