SCHEMBL8329540

SCHEMBL8329540

CCOC(=O)C(CCCNC(=O)OC(C)(C)C)(OCc1ccccc1)C(=O)OCC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.50
SYK P43405 1/20 0.48
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
HDAC9 Q9UKV0 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
NCOR2 Q9Y618 1/20 0.46
HTT P42858 1/20 0.46
MAPT P10636 3/20 0.46
SIGMAR1 Q99720 2/20 0.45
PTPRB P23467 1/20 0.43
L3MBTL1 Q9Y468 3/20 0.43
CYP3A4 P08684 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8803281 0.90 HDAC3 (0.51) IDO1SYKHDAC3HDAC4HDAC1
SCHEMBL8799761 0.89 CYP3A4 (0.44) IDO1SYKMAPTPTPRBCYP3A4
SCHEMBL8799056 0.89 SIGMAR1 (0.51) IDO1SYKHDAC3HDAC4HDAC1
SCHEMBL8798754 0.88 CYP3A4 (0.57) IDO1SYKHDAC3HDAC4HDAC1
SCHEMBL8800029 0.85 KEAP1 (0.42) IDO1MAPTPTPRBL3MBTL1CYP3A4
SCHEMBL8633540 0.83 IDO1 (0.46) IDO1SYKHDAC3HDAC4HDAC1
SCHEMBL8798252 0.81 CYP3A4 (0.56) IDO1HDAC3HDAC4HDAC1HDAC7
SCHEMBL8633439 0.79 NPSR1 (0.46) IDO1SYKMAPTPTPRBCYP3A4
SCHEMBL8331034 0.79 TDP1 (0.44) IDO1HTTPTPRBALDH1A1MEN1
SCHEMBL8800128 0.79 CA12 (0.47) MAPTL3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908863-A ANTIGROWTH AGENT FOR BONES DOMPE' S.P.A. (IT) 1999-06-01 US disclosed
EP-0792878-A2 Geminal carboxylic acids and esters thereof, pharmaceutical formulations containing them useful in the treatment of bone dysmetabolism Dompé S.P.A. (IT) 1997-09-03 EP disclosed