SCHEMBL8330266

SCHEMBL8330266

CCC(=O)N(C)C1CC1c1cc(F)ccc1F

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.46
KDM1B Q8NB78 1/20 0.46
GPR88 Q9GZN0 1/20 0.39
RIPK1 Q13546 2/20 0.37
MAPT P10636 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
OPRM1 P35372 1/20 0.36
FFAR1 O14842 1/20 0.36
HCRTR2 O43614 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8335020 0.89 KDM1A (0.44) KDM1AKDM1BGPR88RIPK1OPRM1
SCHEMBL8329899 0.84 KDM1A (0.50) KDM1AKDM1BGPR88FFAR1
SCHEMBL8330750 0.83 KDM1A (0.46) KDM1AKDM1BGPR88RIPK1FFAR1
SCHEMBL8331376 0.77 MEN1 (0.36) OPRM1
SCHEMBL8333857 0.76 F2R (0.37) OPRM1
SCHEMBL8333635 0.71 HTR2A (0.44)
SCHEMBL8089391 0.70 MTNR1B (0.52) KDM1AKDM1BFFAR1
SCHEMBL8089388 0.70 MTNR1B (0.52) KDM1AKDM1BFFAR1
SCHEMBL23993612 0.69 KDM1A (0.58) KDM1AKDM1BFFAR1
SCHEMBL16591229 0.69 KDM1A (0.58) KDM1AKDM1BFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889031-A CONTROLLING CIRCADIAN RHYTHMS BRISTOL-MYERS SQUIBB COMPNAY (US) 1999-03-30 US disclosed
US-5753709-A N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-19 US disclosed