SCHEMBL8330435

SCHEMBL8330435

CC(=O)N(C)C1CC1c1cccc(Br)c1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.49
HTR2A P28223 5/20 0.43
HTR2C P28335 5/20 0.43
HTR2B P41595 5/20 0.43
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
HRH3 Q9Y5N1 5/20 0.41
MAPT P10636 1/20 0.40
F2RL1 P55085 1/20 0.39
HDAC4 P56524 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8331075 0.85 KDM1A (0.45) KDM1AHTR2AHTR2CHTR2BSLC6A4
SCHEMBL8331070 0.84 HTR2C (0.44) KDM1AHTR2AHTR2CHTR2BSLC6A4
SCHEMBL8332820 0.82 KDM1A (0.43) KDM1AHTR2AHTR2CHTR2BSLC6A4
SCHEMBL8333596 0.82 SLC9A1 (0.47) HTR2AHTR2CHTR2BSLC6A3HRH3
SCHEMBL7002740 0.81 MAOA (0.51) KDM1AHTR2CSLC6A3MAPTHDAC4
SCHEMBL8332789 0.80 SLC9A1 (0.51) HTR2AHTR2CHTR2B
SCHEMBL25606213 0.75 KDM1A (0.54) KDM1AHTR2AHTR2CHTR2BSLC6A4
SCHEMBL6753587 0.75 HTR2A (0.42) KDM1AHTR2AHTR2CHTR2B
SCHEMBL6753585 0.75 HTR2A (0.42) KDM1AHTR2AHTR2CHTR2B
SCHEMBL4134736 0.70 KDM1A (0.56) KDM1AHTR2AHTR2CHTR2BSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889031-A CONTROLLING CIRCADIAN RHYTHMS BRISTOL-MYERS SQUIBB COMPNAY (US) 1999-03-30 US disclosed
US-5753709-A N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-19 US disclosed