SCHEMBL8333598

SCHEMBL8333598

CC(C(N)=O)C1CC1c1cccc(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 2/20 0.52
HTR2A P28223 2/20 0.47
HTR2C P28335 2/20 0.47
HTR2B P41595 2/20 0.47
ALOX5 P09917 1/20 0.44
MDM2 Q00987 6/20 0.42
TP53 P04637 5/20 0.42
GPR88 Q9GZN0 1/20 0.41
SLC6A3 Q01959 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
KDM1A O60341 1/20 0.40
PARP1 P09874 1/20 0.39
TRPM8 Q7Z2W7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8331072 0.84 HTR2C (0.47) SLC9A1HTR2AHTR2CHTR2BALOX5
SCHEMBL8333640 0.83 SLC9A1 (0.50) SLC9A1HTR2AHTR2CHTR2BALOX5
SCHEMBL8330436 0.83 KDM1A (0.51) SLC9A1HTR2AHTR2CHTR2BALOX5
SCHEMBL8332790 0.81 SLC9A1 (0.56) SLC9A1HTR2AHTR2CHTR2BALOX5
SCHEMBL8332794 0.80 SLC9A1 (0.47) SLC9A1HTR2AHTR2CHTR2BALOX5
SCHEMBL23993596 0.80 HTR2A (0.51) SLC9A1HTR2AHTR2CHTR2BMDM2
SCHEMBL27430078 0.79 SLC9A1 (0.56) SLC9A1ALOX5TP53
SCHEMBL24737578 0.74 SLC9A1 (0.71) SLC9A1HTR2AHTR2CHTR2BMDM2
SCHEMBL24737867 0.74 SLC9A1 (0.71) SLC9A1HTR2AHTR2CHTR2BMDM2
SCHEMBL24737580 0.74 SLC9A1 (0.71) SLC9A1HTR2AHTR2CHTR2BMDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889031-A CONTROLLING CIRCADIAN RHYTHMS BRISTOL-MYERS SQUIBB COMPNAY (US) 1999-03-30 US disclosed
US-5753709-A N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-19 US disclosed