SCHEMBL8330436

SCHEMBL8330436

CC(C(N)=O)C1CC1c1cccc(Br)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 4/20 0.51
SLC6A3 Q01959 2/20 0.46
SLC6A4 P31645 1/20 0.46
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
HTR2B P41595 1/20 0.46
ALOX5 P09917 2/20 0.44
HRH3 Q9Y5N1 1/20 0.40
TSHR P16473 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
PARP1 P09874 1/20 0.39
HDAC4 P56524 1/20 0.38
RCOR1 Q9UKL0 1/20 0.37
F2RL1 P55085 1/20 0.36
CHRNA1 P02708 1/20 0.35
CHRNG P07510 1/20 0.35
CHRNB1 P11230 1/20 0.35
CHRNB2 P17787 1/20 0.35
SLC6A2 P23975 1/20 0.35
CHRNB4 P30926 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8331072 0.84 HTR2C (0.47) KDM1ASLC6A3SLC6A4HTR2AHTR2C
SCHEMBL8331076 0.83 KDM1A (0.49) KDM1ASLC6A3SLC6A4HTR2AHTR2C
SCHEMBL8333598 0.83 SLC9A1 (0.52) KDM1ASLC6A3HTR2AHTR2CHTR2B
SCHEMBL8332790 0.81 SLC9A1 (0.56) HTR2AHTR2CHTR2BALOX5TSHR
SCHEMBL8332822 0.80 KDM1A (0.46) KDM1ASLC6A3SLC6A4HTR2AHTR2C
SCHEMBL27430078 0.79 SLC9A1 (0.56) ALOX5TSHRSLC9A1
SCHEMBL4134867 0.74 KDM1A (0.59) KDM1ASLC6A3SLC6A4HTR2AHTR2C
SCHEMBL4134864 0.74 KDM1A (0.59) KDM1ASLC6A3SLC6A4HTR2AHTR2C
SCHEMBL27350337 0.74 KDM1A (0.50) KDM1ASLC6A3SLC6A4HTR2AHTR2C
SCHEMBL25606213 0.71 KDM1A (0.54) KDM1ASLC6A3SLC6A4HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889031-A CONTROLLING CIRCADIAN RHYTHMS BRISTOL-MYERS SQUIBB COMPNAY (US) 1999-03-30 US disclosed
US-5753709-A N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-19 US disclosed