SCHEMBL8333794

SCHEMBL8333794

CC(CCc1ccc2ccccc2c1)C([NH])=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.50
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
HTR2B P41595 1/20 0.46
CES2 O00748 1/20 0.46
SOX18 P35713 1/20 0.46
GRIN2D O15399 1/20 0.44
GRIN2A Q12879 1/20 0.44
GRIN2B Q13224 1/20 0.44
GRIN2C Q14957 1/20 0.44
HDAC1 Q13547 1/20 0.44
CYP2A6 P11509 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
SIGMAR1 Q99720 2/20 0.44
F2 P00734 1/20 0.44
F10 P00742 1/20 0.44
F7 P08709 1/20 0.44
SLC13A5 Q86YT5 1/20 0.43
PDPK1 O15530 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8102861 0.84 HTR2A (0.57) CYP1A2HTR2AHTR2CHTR2BCYP2A6
SCHEMBL2482277 0.78 HTR2A (0.53) CYP1A2HTR2AHTR2CHTR2BCES2
SCHEMBL7900491 0.78 HTR2A (0.53) CYP1A2HTR2AHTR2CHTR2BCES2
SCHEMBL26846103 0.78 HTR2A (0.56) CYP1A2HTR2AHTR2CHTR2BCES2
SCHEMBL20306138 0.75 CYP1A2 (0.50) CYP1A2HTR2AHTR2CHTR2BSOX18
SCHEMBL24851230 0.75 HTR2A (0.53) CYP1A2HTR2AHTR2CHTR2BCES2
SCHEMBL28648389 0.75 HTR2A (0.53) CYP1A2HTR2AHTR2CHTR2BCES2
SCHEMBL27862101 0.74 CYP1A2 (0.57) CYP1A2SOX18HDAC1HDAC8SLC13A5
SCHEMBL18269436 0.74 CYP1A2 (0.57) CYP1A2HTR2AHTR2CHTR2BCES2
SCHEMBL8190010 0.73 SIGMAR1 (0.53) CYP1A2HTR2AHTR2CHTR2BCES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0890101-A4 SELECTIVELY N-ALKYLATED PEPTIDOMIMETIC COMBINATORIAL LIBRARIES AND COMPOUNDS THEREIN TORREY PINES INST (US) 1999-12-08 EP disclosed
EP-0890101-A1 SELECTIVELY N-ALKYLATED PEPTIDOMIMETIC COMBINATORIAL LIBRARIES AND COMPOUNDS THEREIN TORREY PINES INSTITUTE FOR MOLECULAR STUDIES (US) 1999-01-13 EP disclosed
WO-1997033174-A1 SELECTIVELY N-ALKYLATED PEPTIDOMIMETIC COMBINATORIAL LIBRARIES AND COMPOUNDS THEREIN TORREY PINES INSTITUTE FOR MOLECULAR STUDIES (US) 1997-09-12 WO disclosed