SCHEMBL8334151

SCHEMBL8334151

O=C(O)Cc1cc(-c2ccccn2)nc2cc(O)ccc12

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.46
CYP2C9 P11712 4/20 0.45
CYP3A4 P08684 2/20 0.45
METAP1 P53582 2/20 0.45
MAPK1 P28482 2/20 0.44
NPSR1 Q6W5P4 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
DHODH Q02127 1/20 0.42
LCK P06239 1/20 0.42
FYN P06241 1/20 0.42
AKR1B1 P15121 1/20 0.42
GRB2 P62993 1/20 0.42
LMNA P02545 1/20 0.42
CBFB Q13951 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7952415 0.88 CYP2C9 (0.56) ADORA3CYP2C9CYP3A4METAP1MAPK1
SCHEMBL8335283 0.86 NPSR1 (0.51) ADORA3CYP2C9CYP3A4METAP1MAPK1
SCHEMBL8335971 0.86 ADORA3 (0.45) ADORA3CYP2C9CYP3A4METAP1MAPK1
SCHEMBL8334494 0.86 KMT2A (0.48) ADORA3CYP2C9CYP3A4NPSR1TDP1
SCHEMBL8335356 0.86 KDM4E (0.52) ADORA3CYP2C9CYP3A4METAP1NPSR1
SCHEMBL8335315 0.86 ADORA3 (0.45) ADORA3CYP2C9CYP3A4METAP1MAPK1
SCHEMBL8334301 0.84 METAP1 (0.49) ADORA3METAP1NPSR1LMNA
SCHEMBL8338056 0.84 METAP1 (0.48) ADORA3CYP2C9CYP3A4METAP1MAPK1
SCHEMBL8336614 0.74 KDM4E (0.54) ADORA3CYP2C9CYP3A4METAP1MAPK1
SCHEMBL18473272 0.73 ADORA3 (0.52) ADORA3CYP2C9CYP3A4METAP1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5969150-A FLUORESCENT COMPOUNDS FOR MEDICAL DIAGNOSIS, DRUGS AND LABELS OR FUNGICIDES AND VIRICIDES THE ROCKEFELLER UNIVERSITY (US) 1999-10-19 US disclosed