SCHEMBL8335185

SCHEMBL8335185

CS/C(N)=N\c1cc(C)cc(C(=O)O)c1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TPMT P51580 1/20 0.50
NOS1 P29475 10/20 0.44
NOS3 P29474 8/20 0.44
NOS2 P35228 5/20 0.44
HCAR1 Q9BXC0 1/20 0.44
HCAR2 Q8TDS4 1/20 0.40
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
CNR2 P34972 1/20 0.34
DHODH Q02127 2/20 0.34
ALDH1A1 P00352 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
AOC3 Q16853 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6226312 0.84 CA12 (0.47) TPMTNOS1NOS3NOS2HCAR1
SCHEMBL8335518 0.77 NOS1 (0.71) NOS1NOS3NOS2SMN1; SMN2
SCHEMBL31398620 0.76 NOS1 (0.68) NOS1NOS3NOS2CA12CA1
SCHEMBL13979402 0.73 TPMT (0.64) TPMTHCAR1HCAR2CA12CA1
SCHEMBL8334251 0.70 NEU3 (0.44) TPMTNOS1NOS3NOS2CA12
SCHEMBL221684 0.70 TPMT (1.00) TPMTHCAR1HCAR2CA12CA1
SCHEMBL40661 0.70 TPMT (0.89) TPMTHCAR1HCAR2CA12CA1
SCHEMBL12446319 0.70 TPMT (0.64) TPMTHCAR1HCAR2CA12CA1
SCHEMBL27704356 0.69 TPMT (0.70) TPMTHCAR1HCAR2CA12CA1
SCHEMBL26317012 0.68 TRPA1 (0.58) TPMTHCAR1RXRARXRBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004060376-A1 THE R-ISOMER OF BETA AMINO ACID COMPOUNDS AS INTEGRIN RECEPTOR ANTAGONISTS DERIVATIVES PHARMACIA CORPRATION (US) 2004-07-22 WO disclosed