SCHEMBL8335479

SCHEMBL8335479

O=C(NCc1ccc2c(c1)CCO2)c1cc(C(=O)NCc2cccs2)ncn1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 6/20 0.52
HPGD P15428 4/20 0.52
RAB9A P51151 8/20 0.51
NPC1 O15118 6/20 0.50
POLB P06746 2/20 0.50
EGLN1 Q9GZT9 1/20 0.50
AURKA O14965 1/20 0.48
RPS6KB1 P23443 1/20 0.48
CHRM4 P08173 1/20 0.47
MMP13 P45452 3/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
TP53 P04637 1/20 0.45
TSHR P16473 1/20 0.45
HTT P42858 1/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
KDM4E B2RXH2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8358827 0.89 RAB9A (0.61) HPGDRAB9ANPC1POLBEGLN1
SCHEMBL8335113 0.89 SMN1; SMN2 (0.64) SMN1; SMN2HPGDRAB9ANPC1MMP13
SCHEMBL5615885 0.85 RAB9A (0.54) SMN1; SMN2HPGDRAB9ANPC1POLB
SCHEMBL4718511 0.85 RAB9A (0.59) HPGDRAB9ANPC1POLBEGLN1
SCHEMBL5615618 0.85 RAB9A (0.52) HPGDRAB9ANPC1POLBEGLN1
SCHEMBL5616132 0.84 RAB9A (0.49) HPGDRAB9ANPC1POLBEGLN1
SCHEMBL5616113 0.83 RAB9A (0.56) HPGDRAB9ANPC1POLBEGLN1
SCHEMBL5616109 0.83 RAB9A (0.55) HPGDRAB9ANPC1POLBEGLN1
SCHEMBL8360215 0.83 MMP13 (0.69) HPGDRAB9ANPC1POLBEGLN1
SCHEMBL8357430 0.83 RAB9A (0.52) HPGDRAB9ANPC1POLBEGLN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7166609-B2 Pyrimidine-4,6-dicarboxylic acid diamides for selectively inhibiting collagenases SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2007-01-23 US disclosed
US-7166609-B2 Pyrimidine-4,6-dicarboxylic acid diamides for selectively inhibiting collagenases SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2007-01-23 US disclosed
WO-2004041788-A1 NOVEL PYRIMIDINE-4,6-DICARBOXAMIDES FOR THE SELECTIVE INHIBITION OF COLLAGENASES AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2004-05-21 WO disclosed