SCHEMBL8337124

SCHEMBL8337124

CCC(c1ccc(-c2ccc(Br)cc2)cc1)c1c(O)c2ccccc2oc1=O

nearest known ligand 0.77

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 6/20 0.77
THRB P10828 1/20 0.74
NQO1 P15559 3/20 0.64
CTSK P43235 1/20 0.58
VKORC1 Q9BQB6 2/20 0.58
KDM4E B2RXH2 2/20 0.58
ALDH1A1 P00352 1/20 0.58
ALB P02768 1/20 0.58
PCSK7 Q16549 1/20 0.58
HSD17B10 Q99714 1/20 0.58
MEN1 O00255 1/20 0.58
KMT2A Q03164 1/20 0.58
POLB P06746 1/20 0.57
TOP1 P11387 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8332272 0.91 THRB (0.71) CYP2C9THRBNQO1CTSKVKORC1
SCHEMBL8339057 0.89 THRB (0.69) CYP2C9THRBNQO1CTSKVKORC1
SCHEMBL8335244 0.88 THRB (0.78) CYP2C9THRBNQO1CTSKVKORC1
SCHEMBL8333320 0.87 THRB (0.70) CYP2C9THRBNQO1CTSKVKORC1
SCHEMBL8523615 0.87 THRB (0.70) CYP2C9THRBNQO1CTSKVKORC1
Phenprocoumon SCHEMBL24500472 0.87 CYP2C9 (1.00) CYP2C9NQO1VKORC1KDM4EALDH1A1
Phenprocoumon SCHEMBL43031 0.87 CYP2C9 (1.00) CYP2C9NQO1VKORC1KDM4EALDH1A1
Phenprocoumon SCHEMBL24500477 0.87 CYP2C9 (1.00) CYP2C9NQO1VKORC1KDM4EALDH1A1
Phenprocoumon SCHEMBL29392123 0.87 CYP2C9 (1.00) CYP2C9NQO1VKORC1KDM4EALDH1A1
SCHEMBL8334663 0.87 THRB (0.72) CYP2C9THRBNQO1CTSKVKORC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999001446-A1 NOVEL 4-HYDROXY-2H-1-(THIO)PYRAN-2-ONES DERIVATIVES AND THEIR USE AS RAT POISON LIPHATEC (FR) 1999-01-14 WO claimed
WO-1999001446-A1 NOVEL 4-HYDROXY-2H-1-(THIO)PYRAN-2-ONES DERIVATIVES AND THEIR USE AS RAT POISON LIPHATEC (FR) 1999-01-14 WO disclosed