SCHEMBL8333320

SCHEMBL8333320

CC(C)(C)CC(c1ccc(-c2ccc(Br)cc2)cc1)c1c(O)c2ccccc2oc1=O

nearest known ligand 0.70

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.70
NQO1 P15559 3/20 0.60
CYP2C9 P11712 6/20 0.58
CTSK P43235 1/20 0.55
VKORC1 Q9BQB6 3/20 0.55
KDM4E B2RXH2 2/20 0.55
ALB P02768 2/20 0.55
ALDH1A1 P00352 1/20 0.55
PCSK7 Q16549 1/20 0.55
HSD17B10 Q99714 1/20 0.55
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
POLB P06746 1/20 0.54
TOP1 P11387 1/20 0.53
TOP2A P11388 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8337124 0.87 CYP2C9 (0.77) THRBNQO1CYP2C9CTSKVKORC1
SCHEMBL8335244 0.85 THRB (0.78) THRBNQO1CYP2C9CTSKVKORC1
SCHEMBL8332272 0.85 THRB (0.71) THRBNQO1CYP2C9CTSKVKORC1
SCHEMBL8523615 0.84 THRB (0.70) THRBNQO1CYP2C9CTSKVKORC1
SCHEMBL8334663 0.84 THRB (0.72) THRBNQO1CYP2C9CTSKVKORC1
SCHEMBL8339057 0.83 THRB (0.69) THRBNQO1CYP2C9CTSKVKORC1
SCHEMBL8336582 0.82 VKORC1 (0.74) THRBNQO1CYP2C9VKORC1KDM4E
Bromodiolone SCHEMBL433993 0.82 THRB (1.00) THRBNQO1CYP2C9CTSKVKORC1
Bromodiolone SCHEMBL29362860 0.82 THRB (1.00) THRBNQO1CYP2C9CTSKVKORC1
SCHEMBL31398272 0.82 NQO1 (0.62) THRBNQO1CYP2C9VKORC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999001446-A1 NOVEL 4-HYDROXY-2H-1-(THIO)PYRAN-2-ONES DERIVATIVES AND THEIR USE AS RAT POISON LIPHATEC (FR) 1999-01-14 WO disclosed