SCHEMBL8335244

SCHEMBL8335244

CC(C)CC(c1ccc(-c2ccc(Br)cc2)cc1)c1c(O)c2ccccc2oc1=O

nearest known ligand 0.78

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.78
CYP2C9 P11712 7/20 0.65
VKORC1 Q9BQB6 3/20 0.65
NQO1 P15559 4/20 0.61
KDM4E B2RXH2 2/20 0.60
POLB P06746 1/20 0.60
CTSK P43235 1/20 0.56
ALDH1A1 P00352 1/20 0.56
ALB P02768 1/20 0.56
PCSK7 Q16549 1/20 0.56
HSD17B10 Q99714 1/20 0.56
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
CRHBP P24387 1/20 0.55
CASP7 P55210 1/20 0.55
CASP6 P55212 1/20 0.55
CRHR2 Q13324 1/20 0.55
HIF1A Q16665 1/20 0.55
TOP1 P11387 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8523615 0.90 THRB (0.70) THRBCYP2C9VKORC1NQO1KDM4E
SCHEMBL8337124 0.88 CYP2C9 (0.77) THRBCYP2C9VKORC1NQO1KDM4E
SCHEMBL7351597 0.88 CYP2C9 (0.82) THRBCYP2C9VKORC1NQO1KDM4E
Bromodiolone SCHEMBL29362860 0.88 THRB (1.00) THRBCYP2C9VKORC1NQO1KDM4E
Bromodiolone SCHEMBL433993 0.88 THRB (1.00) THRBCYP2C9VKORC1NQO1KDM4E
SCHEMBL8332272 0.86 THRB (0.71) THRBCYP2C9VKORC1NQO1KDM4E
SCHEMBL8336582 0.86 VKORC1 (0.74) THRBCYP2C9VKORC1NQO1KDM4E
SCHEMBL8333320 0.85 THRB (0.70) THRBCYP2C9VKORC1NQO1KDM4E
SCHEMBL8334663 0.85 THRB (0.72) THRBCYP2C9VKORC1NQO1KDM4E
SCHEMBL8339057 0.84 THRB (0.69) THRBCYP2C9VKORC1NQO1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999001446-A1 NOVEL 4-HYDROXY-2H-1-(THIO)PYRAN-2-ONES DERIVATIVES AND THEIR USE AS RAT POISON LIPHATEC (FR) 1999-01-14 WO claimed
WO-1999001446-A1 NOVEL 4-HYDROXY-2H-1-(THIO)PYRAN-2-ONES DERIVATIVES AND THEIR USE AS RAT POISON LIPHATEC (FR) 1999-01-14 WO disclosed