SCHEMBL8338137

SCHEMBL8338137

CC(C(=O)O)c1ccccc1CN1C(=O)c2ccccc2C1=O

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.46
CA12 O43570 1/20 0.46
CA9 Q16790 1/20 0.46
KMT2A Q03164 5/20 0.46
PTGS2 P35354 2/20 0.43
GRM5 P41594 1/20 0.43
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
GAA P10253 1/20 0.42
TSHR P16473 1/20 0.42
CYP2C19 P33261 1/20 0.42
ELANE P08246 1/20 0.42
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8341619 0.99 CASP3 (0.45) CASP3CA12CA9KMT2APTGS2
SCHEMBL23748222 0.78 CASP3 (0.47) CASP3CA12CA9KMT2AGRM5
SCHEMBL5112475 0.76 PTGS2 (0.46) PTGS2CYP3A4ALDH1A1
SCHEMBL5983552 0.76 PTGS2 (0.46) PTGS2CYP3A4ALDH1A1
SCHEMBL30222272 0.76 PTGS2 (0.46) PTGS2CYP3A4ALDH1A1
SCHEMBL23748314 0.75 CASP3 (0.47) CASP3CA12CA9KMT2AGRM5
SCHEMBL3213661 0.74 CASP3 (0.49) CASP3CA12CA9KMT2AGRM5
SCHEMBL7987177 0.74 CASP3 (0.49) CASP3CA12CA9KMT2AGRM5
SCHEMBL7822153 0.74 PTGS2 (0.44) KMT2APTGS2MEN1CYP1A2GAA
SCHEMBL1063487 0.74 PTGS2 (0.44) KMT2APTGS2CYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5902803-A 5H,10H-imidazo 1,2-a!indeno 1,2-e!pyrazin-4-one derivatives, preparation thereof, and drugs containing said derivatives RHONE-POULENC RORER S.A. (FR) 1999-05-11 US disclosed