SCHEMBL8341853

SCHEMBL8341853

C/N=C\c1cc(C)cnc1N

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 2/20 0.50
NOS2 P35228 2/20 0.50
NOS1 P29475 1/20 0.50
CYP2A6 P11509 2/20 0.37
CCR1 P32246 1/20 0.32
CCR5 P51681 1/20 0.32
CCR8 P51685 1/20 0.32
ADRA2A P08913 2/20 0.32
ADRA2B P18089 2/20 0.32
ADRA2C P18825 2/20 0.32
PLAU P00749 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20125043 0.76 NOS3 (0.54) NOS3NOS2NOS1CYP2A6CCR1
SCHEMBL8296665 0.76 NOS3 (0.54) NOS3NOS2NOS1CYP2A6CCR1
SCHEMBL20124974 0.76 NOS3 (0.54) NOS3NOS2NOS1CYP2A6CCR1
SCHEMBL25129348 0.70 NOS3 (0.47) NOS3NOS2NOS1CYP2A6CCR1
SCHEMBL8341793 0.68 SMN1; SMN2 (0.48)
SCHEMBL19258550 0.68 NOS3 (0.43) NOS3NOS2NOS1CYP2A6CCR1
SCHEMBL20721716 0.68 PLAU (0.44) NOS3NOS2NOS1PLAU
SCHEMBL20746021 0.68 PLAU (0.44) NOS3NOS2NOS1PLAU
SCHEMBL31619921 0.68
SCHEMBL172774 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004083174-A2 SULFONYL-AMIDINO CONTAINING AND TETRAHYDROPYRIMIDINO CONTAINING COMPOUNDS AS FACTOR XA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-09-30 WO disclosed