SCHEMBL8343164

SCHEMBL8343164

O=c1[nH]c2cc(C(F)(F)F)ccc2n(CCN2CCOCC2)c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.45
ABCB11 O95342 1/20 0.45
HTR1A P08908 1/20 0.45
ADRA2A P08913 1/20 0.45
ADORA3 P0DMS8 1/20 0.45
CHRM1 P11229 1/20 0.45
DRD1 P21728 1/20 0.45
TBXA2R P21731 1/20 0.45
SLC6A4 P31645 1/20 0.45
ADRA1A P35348 1/20 0.45
OPRM1 P35372 1/20 0.45
DRD3 P35462 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
PDE5A O76074 2/20 0.42
PDE9A O76083 2/20 0.42
PARP1 P09874 1/20 0.42
PLK1 P53350 1/20 0.41
PIK3CD O00329 1/20 0.41
PIK3CB P42338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7478166 0.80 PDE5A (0.50) MEN1KMT2APDE5APDE9A
SCHEMBL8345718 0.80 MEN1 (0.51) MEN1KMT2APDE5APDE9A
SCHEMBL5545647 0.79 HTR7 (0.55) MEN1KMT2APARP1
SCHEMBL24335140 0.78 PDE5A (0.48) MEN1KMT2APDE5APDE9APLK1
SCHEMBL29580737 0.78 PDE5A (0.48) MEN1KMT2APDE5APDE9APLK1
SCHEMBL8117343 0.78 MEN1 (0.47) MEN1KMT2APDE5APDE9ARAB9A
SCHEMBL9544064 0.77 GRIA1 (0.55) MEN1KMT2APDE5APDE9A
SCHEMBL8346269 0.77 MEN1 (0.46) MEN1KMT2APDE5APDE9ARAB9A
SCHEMBL13801880 0.76 HTR7 (0.47) KCNH2ABCB11HTR1AADRA2AADORA3
SCHEMBL8118534 0.75 MEN1 (0.45) KCNH2ABCB11HTR1AADRA2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5955461-A Quinoxalinedione derivatives, their production and use in pharmaceutical agents SCHERING AKTIENGESELLSCHAFT (DE) 1999-09-21 US disclosed
US-5750525-A Quinoxalinedione derivatives, their production and use in pharmaceutical agents SCHERING AKTIENGESELLSCHAFT (DE) 1998-05-12 US disclosed