SCHEMBL8344288

SCHEMBL8344288

CC(C)(C)CN(Cc1ccc(C#CCCl)cc1)c1ccnc(N)n1

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GPR4 P46093 7/20 0.52
CTSK P43235 13/20 0.52
HRH3 Q9Y5N1 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8344239 0.89 CTSK (0.52) GPR4CTSKHRH3
SCHEMBL3451101 0.84 CTSK (0.71) GPR4CTSK
SCHEMBL8348852 0.84 GPR4 (0.40) GPR4CTSKHRH3
SCHEMBL8344106 0.83 CTSK (0.51) GPR4CTSKHRH3
SCHEMBL8344244 0.80 CTSK (0.52) GPR4CTSKHRH3
SCHEMBL8344278 0.79 CTSK (0.67) GPR4CTSKHRH3
SCHEMBL8344410 0.78 CTSK (0.79) GPR4CTSK
SCHEMBL8344109 0.77 GPR4 (0.52) GPR4CTSKHRH3
SCHEMBL8346972 0.77 CTSK (0.59) GPR4CTSK
SCHEMBL8345986 0.76 CTSK (0.46) GPR4CTSKHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537111-B1 HETEREOARYL NITRILE DERIVATIVES NOVARTIS AG (CH) 2007-05-02 EP disclosed
WO-2004020441-A1 HETEREOARYL NITRILE DERIVATIVES NOVARTIS AG (CH) 2004-03-11 WO disclosed