SCHEMBL8346972

SCHEMBL8346972

CC(C)(C)CN(Cc1ccc(C#CCN2CCC(C(=O)O)CC2)cc1)c1ccnc(N)n1

nearest known ligand 0.59

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CTSK P43235 10/20 0.59
GPR4 P46093 9/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8346982 0.91 CTSK (0.57) CTSKGPR4
SCHEMBL3450766 0.88 CTSK (0.77) CTSKGPR4
SCHEMBL8344239 0.81 CTSK (0.52) CTSKGPR4
SCHEMBL13109183 0.77 CTSK (0.68) CTSKGPR4
SCHEMBL8344288 0.77 GPR4 (0.52) CTSKGPR4
SCHEMBL3915160 0.76 CTSK (0.77) CTSKGPR4
SCHEMBL13124829 0.76 CTSK (0.60) CTSKGPR4
SCHEMBL8344106 0.74 CTSK (0.51) CTSKGPR4
SCHEMBL8347898 0.73 CTSK (0.59) CTSKGPR4
SCHEMBL3451415 0.71 CTSK (0.78) CTSKGPR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537111-B1 HETEREOARYL NITRILE DERIVATIVES NOVARTIS AG (CH) 2007-05-02 EP disclosed
WO-2004020441-A1 HETEREOARYL NITRILE DERIVATIVES NOVARTIS AG (CH) 2004-03-11 WO disclosed