SCHEMBL8345374

SCHEMBL8345374

CN1C(=O)C(Cc2ccc([S+](C)[O-])cc2)Cc2cc(C(=O)NCc3ccc(C#N)cc3)cnc21

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RORC P51449 6/20 0.44
CXCR3 P49682 2/20 0.42
ROCK2 O75116 2/20 0.40
KDM1A O60341 1/20 0.38
HDAC1 Q13547 1/20 0.38
PRKAA2 P54646 4/20 0.38
EPHX2 P34913 1/20 0.38
ROCK1 Q13464 1/20 0.37
EGLN2 Q96KS0 1/20 0.37
TP53 P04637 1/20 0.37
DRD2 P14416 2/20 0.36
DRD3 P35462 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6748396 0.74 SMN1; SMN2 (0.43) RORCCXCR3ROCK2PRKAA2TP53
SCHEMBL20903790 0.67 RORC (0.56) RORC
SCHEMBL19864642 0.64 TP53 (0.45) ROCK2KDM1AHDAC1EPHX2ROCK1
SCHEMBL19864600 0.63 TP53 (0.44) ROCK2EPHX2ROCK1TP53DRD2
SCHEMBL19864629 0.63 LMNA (0.44) HDAC1EPHX2
SCHEMBL7445367 0.62 ITGB3 (0.54)
SCHEMBL7445376 0.62 ITGB3 (0.54)
SCHEMBL21277705 0.62 RORC (0.51) RORCCXCR3ROCK2KDM1AHDAC1
SCHEMBL21277672 0.62 RORC (0.58) RORC
SCHEMBL18745170 0.61 RORC (1.00) RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014389-A1 3,4-DIHYDROQUINOLIN-2-ONE, 5,6-FUSED OXAZIN-3-ONE, AND 5,6-FUSED THIAZIN-3-ONE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed