SCHEMBL8345768

SCHEMBL8345768

CC(CO)c1ccc(CN(CC(C)(C)C)c2ccnc(N)n2)cc1

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSK P43235 11/20 0.46
GPR4 P46093 7/20 0.40
HRH3 Q9Y5N1 2/20 0.37
HRH4 Q9H3N8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3451762 0.83 CTSK (0.69) CTSKGPR4
SCHEMBL14528153 0.83 HRH4 (0.41) CTSKGPR4HRH4
SCHEMBL8345765 0.83 CTSK (0.45) CTSKGPR4HRH3HRH4
SCHEMBL8344244 0.81 CTSK (0.52) CTSKGPR4HRH3HRH4
SCHEMBL8345749 0.81 CTSK (0.47) CTSKGPR4HRH3
SCHEMBL8344278 0.80 CTSK (0.67) CTSKGPR4HRH3
SCHEMBL8346784 0.78 GPR4 (0.48) CTSKGPR4HRH3
SCHEMBL8344239 0.78 CTSK (0.52) CTSKGPR4HRH3
SCHEMBL8344106 0.77 CTSK (0.51) CTSKGPR4HRH3
SCHEMBL8344288 0.74 GPR4 (0.52) CTSKGPR4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537111-B1 HETEREOARYL NITRILE DERIVATIVES NOVARTIS AG (CH) 2007-05-02 EP disclosed
WO-2004020441-A1 HETEREOARYL NITRILE DERIVATIVES NOVARTIS AG (CH) 2004-03-11 WO disclosed