SCHEMBL8345848

SCHEMBL8345848

Cc1ccc(C)c(NC(=O)C(NC(=O)OC(C)(C)C)c2ccccc2)c1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.56
CTSK P43235 1/20 0.56
BRD4 O60885 1/20 0.51
ALDH1A1 P00352 3/20 0.49
KMT2A Q03164 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.46
MAPT P10636 3/20 0.46
LMNA P02545 3/20 0.45
THRB P10828 1/20 0.45
TP53 P04637 1/20 0.45
S1PR3 Q99500 1/20 0.45
MEN1 O00255 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8334464 0.91 CTSS (0.56) CTSSCTSKALDH1A1KMT2ASMN1; SMN2
SCHEMBL8348046 0.89 CTSS (0.54) CTSSCTSKSMN1; SMN2MAPTS1PR3
SCHEMBL8348878 0.89 CTSS (0.54) CTSSCTSKALDH1A1KMT2ASMN1; SMN2
SCHEMBL8337352 0.88 CTSS (0.60) CTSSCTSKALDH1A1SMN1; SMN2MAPT
SCHEMBL8348009 0.88 CTSS (0.60) CTSSCTSKALDH1A1SMN1; SMN2MAPT
SCHEMBL6824801 0.85 BRD4 (0.60) BRD4ALDH1A1KMT2ASMN1; SMN2MAPT
SCHEMBL8336332 0.83 CTSS (0.60) CTSSCTSKALDH1A1KMT2ASMN1; SMN2
SCHEMBL8336972 0.82 CTSS (0.57) CTSSCTSKALDH1A1MAPTTP53
SCHEMBL8336805 0.82 CTSS (0.57) CTSSCTSKKMT2AMAPTTHRB
SCHEMBL8337969 0.82 CTSS (0.57) CTSSCTSKALDH1A1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004022534-A1 ARYLGLYCINE DERIVATIVES FOR USE AS GLYCINE TRANSPORT INHIBITORS NPS ALLELIX CORP. (CA) 2004-03-18 WO disclosed