SCHEMBL8345990

SCHEMBL8345990

CC(C)(C)OC(=O)NCCCC[C@H](NC(=O)[C@H]1O[C@@H]1C(=O)NCCc1ccccc1)C(=O)Nc1cccc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
CTSK P43235 2/20 0.44
CXCR3 P49682 3/20 0.44
MMP1 P03956 1/20 0.43
MMP3 P08254 1/20 0.43
MMP9 P14780 1/20 0.43
KLK7 P49862 2/20 0.43
KLK5 Q9Y337 2/20 0.43
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
MAPT P10636 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CTSS P25774 1/20 0.41
SIRT5 Q9NXA8 1/20 0.40
PAX8 Q06710 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8349352 0.91 CA1 (0.47) CA1CA2CTSKCXCR3KLK7
SCHEMBL8345432 0.86 HDAC1 (0.51) HDAC1HDAC2SIRT5
SCHEMBL8346795 0.85 KDM4E (0.45) CA1CA2CXCR3KLK7KLK5
SCHEMBL8349391 0.85 NTMT1 (0.51) CA1CA2MMP1MMP3MMP9
SCHEMBL7764063 0.85 NTMT1 (0.51) CA1CA2MMP1MMP3MMP9
Hydrochloric Acid SCHEMBL7759028 0.85 NTMT1 (0.51) CA1CA2MMP1MMP3MMP9
Hydrochloric Acid SCHEMBL8344064 0.85 NTMT1 (0.51) CA1CA2MMP1MMP3MMP9
Hydrochloric Acid SCHEMBL8342864 0.82 NTMT1 (0.50) MMP1MMP3MMP9HDAC1HDAC2
Hydrochloric Acid SCHEMBL7764068 0.82 NTMT1 (0.50) MMP1MMP3MMP9HDAC1HDAC2
SCHEMBL8349755 0.81 HDAC1 (0.50) HDAC1HDAC2SIRT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5883121-A INHIBITING ACTIVITY AGAINST CATHEPSIN, AND IS USEFUL FOR PREVENTION AND TREATMENT OF OSTEOPATHY SUCH AS OSTEOPOROSIS TAIHO PHARMACEUTICAL CO., LTD. (JP) 1999-03-16 US disclosed