SCHEMBL8349352

SCHEMBL8349352

CC(C)(C)OC(=O)NCCCC[C@H](NC(=O)[C@H]1O[C@@H]1C(=O)Nc1cccc2ccccc12)C(=O)Nc1cccc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.47
CA2 P00918 3/20 0.47
HSD17B10 Q99714 1/20 0.43
CXCR3 P49682 1/20 0.42
ALDH1A1 P00352 1/20 0.42
SIRT5 Q9NXA8 1/20 0.42
NTMT1 Q9BV86 1/20 0.42
HDAC1 Q13547 4/20 0.41
HDAC4 P56524 3/20 0.41
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
KLK7 P49862 1/20 0.40
KLK5 Q9Y337 1/20 0.40
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC3 O15379 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC10 Q969S8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8345990 0.91 CA1 (0.46) CA1CA2CXCR3SIRT5HDAC1
SCHEMBL8346795 0.91 KDM4E (0.45) CA1CA2HSD17B10CXCR3NTMT1
SCHEMBL7759044 0.81 NTMT1 (0.58) HSD17B10NTMT1HDAC1HDAC4HDAC2
SCHEMBL8343138 0.81 NTMT1 (0.58) HSD17B10NTMT1HDAC1HDAC4HDAC2
Hydrochloric Acid SCHEMBL7763503 0.81 NTMT1 (0.57) HSD17B10NTMT1HDAC1HDAC4HDAC2
Hydrochloric Acid SCHEMBL8349180 0.81 NTMT1 (0.57) HSD17B10NTMT1HDAC1HDAC4HDAC2
SCHEMBL7762702 0.80 ALDH1A1 (0.49) CA1CA2HSD17B10ALDH1A1CTSS
SCHEMBL8345432 0.79 HDAC1 (0.51) SIRT5HDAC1HDAC4HDAC2HDAC3
SCHEMBL8349755 0.79 HDAC1 (0.50) SIRT5HDAC1HDAC4HDAC2HDAC3
SCHEMBL8349145 0.78 HDAC1 (0.49) SIRT5HDAC1HDAC4HDAC2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5883121-A INHIBITING ACTIVITY AGAINST CATHEPSIN, AND IS USEFUL FOR PREVENTION AND TREATMENT OF OSTEOPATHY SUCH AS OSTEOPOROSIS TAIHO PHARMACEUTICAL CO., LTD. (JP) 1999-03-16 US disclosed