SCHEMBL8346167

SCHEMBL8346167

CNS(=O)(=O)c1ccccc1-n1cccc1-c1ccc(F)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.50
PTGS1 P23219 1/20 0.47
CYP1A2 P05177 1/20 0.36
ALOX5AP P20292 5/20 0.36
FEN1 P39748 5/20 0.36
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.34
TP53 P04637 1/20 0.34
GAA P10253 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
HSD17B10 Q99714 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MMP1 P03956 1/20 0.33
MMP2 P08253 1/20 0.33
MMP3 P08254 1/20 0.33
MMP9 P14780 1/20 0.33
MMP12 P39900 1/20 0.33
MMP13 P45452 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8502568 0.82 PTGS2 (0.60) PTGS2PTGS1
SCHEMBL5071002 0.77 PTGS2 (0.73) PTGS2PTGS1ALDH1A1GAATSHR
SCHEMBL8346365 0.72 PTGS2 (0.56) PTGS2PTGS1
SCHEMBL15366568 0.72 FEN1 (0.54) PTGS2PTGS1ALOX5APFEN1ALDH1A1
SCHEMBL8346170 0.72 KMT2A (0.38) PTGS2ALOX5APFEN1ALDH1A1KDM4E
SCHEMBL8505598 0.71 PTGS2 (0.44) PTGS2PTGS1
SCHEMBL7144222 0.71 MAPK14 (0.62)
SCHEMBL8503394 0.70 PTGS1 (0.44) PTGS2PTGS1
SCHEMBL8505063 0.69 PTGS2 (0.44) PTGS2PTGS1
SCHEMBL8505856 0.69 CA2 (0.44) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5932598-A NOVEL SUBSTITUTED SULFONAMIDE COMPOUNDS USEFUL AS PRODRUGS; ADMINISTERING TO TREAT INFLAMMATION-ASSOCIATED PAIN DUE TO CANCER, DENTAL PAIN; CYCLOOXYGENASE-2 INHIBITORS G. D. SEARLE & CO. (US) 1999-08-03 US disclosed