SCHEMBL8346170

SCHEMBL8346170

CNS(=O)(=O)c1cccc(-n2cccc2)c1-c1ccc(F)cc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.38
ALDH1A1 P00352 3/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
PKM P14618 1/20 0.38
LMNA P02545 2/20 0.36
GAA P10253 2/20 0.36
PTGS2 P35354 1/20 0.36
CYP19A1 P11511 1/20 0.34
ALOX5AP P20292 4/20 0.34
FEN1 P39748 4/20 0.34
TDP1 Q9NUW8 1/20 0.33
HSD11B1 P28845 1/20 0.33
TSHR P16473 1/20 0.33
PTGES2 Q9H7Z7 1/20 0.32
GRM5 P41594 1/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8346167 0.72 PTGS2 (0.50) ALDH1A1GAAPTGS2ALOX5APFEN1
SCHEMBL15366568 0.70 FEN1 (0.54) ALDH1A1PTGS2ALOX5APFEN1HSD11B1
SCHEMBL8346365 0.64 PTGS2 (0.56) PTGS2
SCHEMBL9908753 0.63 PKM (0.64) KMT2AALDH1A1MEN1MAPTPKM
SCHEMBL791010 0.62 PTGES2 (0.54) ALDH1A1LMNAALOX5APFEN1TSHR
SCHEMBL8344047 0.62 PTGS2 (0.51) PTGS2ALOX5APFEN1
SCHEMBL4731653 0.62 CYP1A2 (0.55) ALDH1A1LMNAGAAALOX5APFEN1
SCHEMBL1621373 0.62 ALDH1A1 (0.67) KMT2AALDH1A1MAPTGAAALOX5AP
SCHEMBL29689413 0.61 SLC40A1 (0.51) KMT2AALDH1A1LMNAGAAALOX5AP
SCHEMBL4860115 0.61 PTGS2 (0.57) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5932598-A NOVEL SUBSTITUTED SULFONAMIDE COMPOUNDS USEFUL AS PRODRUGS; ADMINISTERING TO TREAT INFLAMMATION-ASSOCIATED PAIN DUE TO CANCER, DENTAL PAIN; CYCLOOXYGENASE-2 INHIBITORS G. D. SEARLE & CO. (US) 1999-08-03 US disclosed