SCHEMBL8346922

SCHEMBL8346922

CN1CCN(Cc2ccc(OCc3cnc(C#N)nc3NC3CCCCC3)cc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSS P25774 10/20 0.52
CTSL P07711 9/20 0.52
CTSK P43235 8/20 0.52
NPC1 O15118 2/20 0.43
TP53 P04637 2/20 0.43
RAB9A P51151 2/20 0.43
CTSB P07858 1/20 0.42
HRH3 Q9Y5N1 3/20 0.42
NSD2 O96028 2/20 0.42
KDM4E B2RXH2 1/20 0.41
AXL P30530 1/20 0.41
FLT3 P36888 1/20 0.41
TYRO3 Q06418 1/20 0.41
MERTK Q12866 1/20 0.41
EHMT2 Q96KQ7 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3451217 0.84 CTSS (0.52) CTSSCTSLCTSKCTSBHRH3
SCHEMBL4141262 0.76 CTSS (0.81) CTSSCTSLCTSK
SCHEMBL13125019 0.72 FLT3 (0.42) CTSSCTSLCTSKNPC1TP53
SCHEMBL3450506 0.69 NSD2 (0.56) CTSSCTSLCTSKNSD2EHMT2
SCHEMBL3451071 0.69 CTSL (0.48) CTSSCTSLCTSKCTSBNSD2
SCHEMBL16231116 0.68 CTSS (1.00) CTSSCTSLCTSKTYRO3
SCHEMBL13125004 0.68 CTSS (0.63) CTSSCTSLCTSKCTSB
SCHEMBL4138661 0.68 CTSK (0.67) CTSSCTSLCTSK
SCHEMBL4141268 0.68 CTSS (0.57) CTSSCTSLCTSKNPC1TP53
SCHEMBL16231117 0.67 CTSS (1.00) CTSSCTSLCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004020441-A1 HETEREOARYL NITRILE DERIVATIVES NOVARTIS AG (CH) 2004-03-11 WO disclosed