SCHEMBL8349489

SCHEMBL8349489

O=C(NCc1ccncc1)c1cc(C(=O)NCc2ccc(F)c(Cl)c2)ncn1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 6/20 0.62
MMP10 P09238 1/20 0.50
MMP9 P14780 1/20 0.50
MMP8 P22894 1/20 0.50
HPGD P15428 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
HSD17B10 Q99714 1/20 0.48
HDAC3 O15379 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
ANO1 Q5XXA6 1/20 0.47
NAMPT P43490 1/20 0.45
MAPK1 P28482 2/20 0.45
KDM4E B2RXH2 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6479481 0.93 MMP13 (0.71) MMP13MMP10MMP9MMP8HPGD
SCHEMBL14256100 0.90 MMP13 (0.65) MMP13MMP10MMP9MMP8HPGD
SCHEMBL8348565 0.89 MMP13 (0.61) MMP13MMP10MMP9MMP8HPGD
SCHEMBL8357429 0.89 MMP13 (0.71) MMP13MMP10MMP9MMP8SMN1; SMN2
SCHEMBL8357432 0.89 MMP13 (0.67) MMP13MMP10MMP9MMP8HPGD
SCHEMBL14448540 0.88 MMP13 (0.65) MMP13MMP10MMP9MMP8HPGD
SCHEMBL8348345 0.86 MMP13 (0.62) MMP13MMP10MMP9MMP8HPGD
SCHEMBL5615854 0.86 MMP13 (0.86) MMP13MMP10MMP9MMP8HPGD
SCHEMBL8360133 0.85 MMP13 (0.62) MMP13MMP10MMP9MMP8HPGD
SCHEMBL14284141 0.85 MMP13 (0.65) MMP13MMP10MMP9MMP8HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004060883-A1 PYRIMIDINE-4,6-DICARBOXYLIC ACID DIAMIDES FOR USE AS SELECTIVE MMP 13 INHIBITORS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2004-07-22 WO disclosed