SCHEMBL8352425

SCHEMBL8352425

Fc1ccc(C(Cl)c2ccc(F)c(F)c2)cc1F

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.44
CES1 P23141 2/20 0.44
NFE2L2 Q16236 2/20 0.34
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
HIF1A Q16665 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MAOB P27338 1/20 0.33
PDPK1 O15530 1/20 0.33
APP P05067 2/20 0.33
MME P08473 1/20 0.32
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
ADAM17 P78536 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4183395 0.80 CES2 (0.41) CES2CES1NFE2L2TSHRPDPK1
SCHEMBL6933110 0.78 CES2 (0.47) CES2CES1NFE2L2PDPK1MME
SCHEMBL28193191 0.76 CES2 (0.45) CES2CES1TSHRPDPK1APP
SCHEMBL26674208 0.75 CES2 (0.42) CES2CES1TSHRPDPK1APP
SCHEMBL247899 0.75 CES2 (0.42) CES2CES1NFE2L2PDPK1APP
SCHEMBL25351287 0.75 SHBG (0.41) CES2CES1TSHRMAPK1TDP1
SCHEMBL20495193 0.75 CES2 (0.42) CES2CES1NFE2L2PDPK1APP
SCHEMBL15011402 0.75 CES2 (0.42) CES2CES1TSHRPDPK1APP
SCHEMBL84476 0.74 LMNA (0.44) CES2CES1NFE2L2TSHRHIF1A
SCHEMBL3897101 0.74 CES2 (0.53) CES2CES1PDPK1MMEAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004031148-A1 PIPERAZINE AND PIPERIDINE DERIVATIVES FOR TREATMENT OF NEUROLOGICAL DISEASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2004-04-15 WO disclosed