SCHEMBL8356552

SCHEMBL8356552

O=c1c2ccccc2sn1CCO

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 4/20 0.66
KAT2A Q92830 2/20 0.65
KAT2B Q92831 2/20 0.65
FAAH O00519 1/20 0.62
MGLL Q99685 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11278746 0.89 CASP3 (0.74) CASP3KAT2AKAT2BFAAHMGLL
SCHEMBL17372961 0.88 FAAH (0.70) CASP3KAT2AKAT2BFAAHMGLL
SCHEMBL11276670 0.87 FAAH (0.73) CASP3KAT2AKAT2BFAAHMGLL
SCHEMBL24836231 0.85 FAAH (0.81) CASP3KAT2AKAT2BFAAHMGLL
SCHEMBL2963555 0.85 CASP3 (0.68) CASP3KAT2AKAT2BFAAHMGLL
SCHEMBL24836229 0.85 FAAH (0.76) CASP3KAT2AKAT2BFAAHMGLL
SCHEMBL24836228 0.84 FAAH (0.84) CASP3KAT2AKAT2BFAAHMGLL
SCHEMBL24690027 0.82 CASP3 (0.66) CASP3KAT2AKAT2BFAAHMGLL
SCHEMBL8070856 0.82 CASP3 (0.66) CASP3KAT2AKAT2BFAAHMGLL
SCHEMBL9376161 0.82 CASP3 (0.66) CASP3KAT2AKAT2BFAAHMGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-11116559-A None JP disclosed
JP-H11116559-A ISOTHIAZOLE DERIVATIVE AND ITS PRODUCTION SUMITOMO SEIKA CHEM CO LTD 1999-04-27 JP disclosed
EP-0625978-A1 PIPERAZINE AND PIPERIDINE DERIVATIVES, AND THEIR USE AS ANTIPSYCHOTICS THE WELLCOME FOUNDATION LIMITED (GB) 1994-11-30 EP disclosed
WO-1993016073-A1 PIPERAZINE AND PIPERIDINE DERIVATIVES, AND THEIR USE AS ANTIPSYCHOTICS THE WELLCOME FOUNDATION LIMITED (GB) 1993-08-19 WO disclosed
EP-0018100-B1 SUBSTITUTED AROMATIC BIOLOGICALLY ACTIVE COMPOUND, A PROCESS FOR ITS PREPARATION AND ITS USE AS BIOCIDE IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1984-01-18 EP disclosed
EP-0018100-A2 Substituted aromatic biologically active compound, a process for its preparation and its use as biocide IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1980-10-29 EP disclosed