SCHEMBL8357933

SCHEMBL8357933

CCN(CCO)CCOc1ccc2sc(Cc3ccc(Cl)cc3)nc2c1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.56
LMNA P02545 1/20 0.43
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 2/20 0.42
AGER Q15109 6/20 0.40
EBP Q15125 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
ATP4A P20648 1/20 0.40
ATP4B P51164 1/20 0.40
ACHE P22303 1/20 0.40
LTA4H P09960 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
AURKB Q96GD4 1/20 0.39
LSS P48449 2/20 0.38
LOXL2 Q9Y4K0 1/20 0.36
CSNK1D P48730 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8359651 0.93 HTT (0.64) HTTLMNACYP1A2CYP2D6AGER
SCHEMBL8361490 0.92 LMNA (0.53) HTTLMNACYP1A2CYP2D6AGER
SCHEMBL8361945 0.87 LMNA (0.51) HTTLMNACYP1A2CYP2D6AGER
SCHEMBL8356218 0.85 LMNA (0.60) HTTLMNACYP1A2CYP2D6AGER
SCHEMBL8359567 0.83 AURKB (0.45) HTTLMNACYP1A2CYP2D6ATP4A
SCHEMBL8552900 0.82 LMNA (0.53) HTTLMNACYP1A2CYP2D6LTA4H
SCHEMBL8357762 0.81 LMNA (0.49) HTTLMNACYP1A2CYP2D6ACHE
SCHEMBL8358021 0.81 HTT (0.44) HTTATP4AATP4BLOXL2
SCHEMBL8551252 0.80 LMNA (0.50) HTTLMNACYP1A2CYP2D6ATP4A
SCHEMBL8355859 0.80 AURKB (0.49) HTTLMNACYP1A2CYP2D6AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919807-A ANTICHOLESTEROL AGENTS DR. KARL THOMAE GMBH (DE) 1999-07-06 US disclosed
EP-0824529-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-02-25 EP disclosed
WO-1996035681-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-11-14 WO disclosed