SCHEMBL8551252

SCHEMBL8551252

CCN(CCO)CCOc1ccc2nc(Cc3ccc(C(F)(F)F)cc3)sc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.50
CYP1A2 P05177 2/20 0.49
CYP2D6 P10635 2/20 0.49
CACNA1B Q00975 4/20 0.44
CACNA1H O95180 1/20 0.44
MAPT P10636 2/20 0.42
LSS P48449 2/20 0.41
CNR2 P34972 2/20 0.40
PPARG P37231 1/20 0.39
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
HTT P42858 2/20 0.38
CSNK1D P48730 1/20 0.38
LTA4H P09960 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA4 P22748 1/20 0.37
ATP4A P20648 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551381 0.94 CACNA1B (0.45) LMNACYP1A2CYP2D6CACNA1BCACNA1H
SCHEMBL8552900 0.90 LMNA (0.53) LMNACYP1A2CYP2D6CACNA1BMAPT
SCHEMBL8551665 0.89 CACNA1B (0.47) LMNACYP1A2CYP2D6CACNA1BCACNA1H
SCHEMBL8554328 0.88 LMNA (0.48) LMNACYP1A2CYP2D6CACNA1BCACNA1H
SCHEMBL8361490 0.88 LMNA (0.53) LMNACYP1A2CYP2D6MAPTLSS
SCHEMBL8359111 0.85 CACNA1B (0.53) LMNACYP1A2CYP2D6CACNA1BCACNA1H
SCHEMBL8359973 0.82 LMNA (0.60) LMNACYP1A2CYP2D6CACNA1BMAPT
SCHEMBL8361945 0.82 LMNA (0.51) LMNACYP1A2CYP2D6LSSHTT
SCHEMBL8516569 0.82 MAPT (0.44) LMNACYP1A2CYP2D6CACNA1BCACNA1H
SCHEMBL8358041 0.82 KMT2A (0.52) LMNACYP1A2CYP2D6MAPTCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0824529-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-02-25 EP disclosed
WO-1996035681-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-11-14 WO disclosed