SCHEMBL8358367

SCHEMBL8358367

CCOC(=O)OC(C)OC(=O)[C@H]1[C@@H]2CC[C@@](N)(C(=O)OC(C)OC(=O)OCC)[C@@H]21

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM8 O00222 1/20 0.40
GRM6 O15303 1/20 0.40
GRM2 Q14416 1/20 0.40
GRM3 Q14832 1/20 0.40
SLC1A2 P43004 1/20 0.38
SLC1A1 P43005 1/20 0.38
CYP3A4 P08684 2/20 0.31
OPRK1 P41145 1/20 0.31
KDM4E B2RXH2 1/20 0.31
THRB P10828 1/20 0.31
HPGD P15428 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8358688 0.86 SLC1A2 (0.40) GRM8GRM6GRM2GRM3SLC1A2
Hydrochloric Acid SCHEMBL6703472 0.81 SLC1A2 (0.36) GRM8GRM6GRM2GRM3SLC1A2
SCHEMBL5690924 0.78 SLC1A2 (0.46) GRM8GRM6GRM2GRM3SLC1A2
SCHEMBL8358427 0.78 MEN1 (0.34) TSHR
Hydrochloric Acid SCHEMBL6703583 0.76 GRM8 (0.41) GRM8GRM6GRM2GRM3SLC1A2
SCHEMBL8354012 0.75 SLC1A2 (0.42) GRM8GRM6GRM2GRM3SLC1A2
SCHEMBL23718843 0.75 SLC1A2 (0.57) GRM8GRM6GRM2GRM3SLC1A2
Hydrochloric Acid SCHEMBL6702822 0.74 SLC1A2 (0.38) GRM8GRM6GRM2GRM3SLC1A2
SCHEMBL6701165 0.72 GRM8 (0.50) GRM8GRM6GRM2GRM3SLC1A2
SCHEMBL8532802 0.70 SLC1A2 (0.44) GRM8GRM6GRM2GRM3SLC1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003045898-A1 PRODRUGS OF EXCITATORY AMINO ACIDS ELI LILLY AND COMPANY (US) 2003-06-05 WO disclosed