SCHEMBL8358490

SCHEMBL8358490

C=CCOc1cc(N)c(F)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPOX P50336 6/20 0.48
HTR2C P28335 13/20 0.46
HTR2B P41595 9/20 0.46
HTR2A P28223 8/20 0.41
ADRB2 P07550 2/20 0.41
HTR1A P08908 2/20 0.41
CHRM5 P08912 2/20 0.41
ADRA2A P08913 2/20 0.41
DRD2 P14416 2/20 0.41
ADRA2B P18089 2/20 0.41
ADRA2C P18825 2/20 0.41
DRD4 P21917 2/20 0.41
HRH2 P25021 2/20 0.41
SLC6A4 P31645 2/20 0.41
HTR7 P34969 2/20 0.41
DRD3 P35462 2/20 0.41
HTR6 P50406 2/20 0.41
KCNH2 Q12809 2/20 0.41
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9781225 0.84 NPC1 (0.50) PPOXHTR2CHTR2BHTR2AADRA2A
SCHEMBL8599856 0.81 NPC1 (0.36) PPOXHTR2CHTR2BGAA
SCHEMBL8599861 0.81 NPC1 (0.36) PPOXHTR2CHTR2BGAA
SCHEMBL8601896 0.81 NPC1 (0.36) PPOXHTR2CHTR2BGAA
SCHEMBL7887159 0.80 HTR2C (0.41) PPOXHTR2CHTR2BHTR2AADRB2
SCHEMBL8177207 0.80 PPOX (0.45) PPOXHTR2CHTR2BHTR2AADRB2
SCHEMBL6408609 0.80 ADRA2A (0.40) PPOXADRA2AADRA2BADRA2CGAA
SCHEMBL30826270 0.79 HTR2C (0.48) PPOXHTR2CHTR2BHTR2AADRB2
SCHEMBL9873406 0.78 PPOX (0.44) PPOXHTR2CHTR2BHTR2AADRB2
SCHEMBL9873396 0.78 NPC1 (0.36) PPOXGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113200924-B 4-amino-5-pyrimidine formamide compound and preparation method and application thereof 南开大学 2022-11-01 CN disclosed
CN-113200985-B Pteridinone compound and preparation method and application thereof 南开大学 2022-09-09 CN disclosed
CN-113200924-A 4-amino-5-pyrimidine formamide compound and preparation method and application thereof 南开大学 2021-08-03 CN disclosed
CN-113200985-A Pteridinone compound and preparation method and application thereof 南开大学 2021-08-03 CN disclosed
EP-0763011-B1 PROCESS FOR THE PREPARATION OF UNSATURATED AMINO COMPOUNDS NOVARTIS AG (CH) 1999-12-29 EP disclosed
US-5856578-A CATALYTIC HYDROGENATION OF THE CORRESPONDING AROMATIC NITRO COMPOUND IN PRESENCE OF NOBLE METAL CATALYST NORVARTIS CORPORATION (US) 1999-01-05 US disclosed
EP-0626370-B1 Process for producing aromatic isothiocyanate derivatives SUMITOMO CHEMICAL CO (JP) 1998-02-11 EP disclosed
US-5631209-A ALGICIDES ROHM AND HAAS COMPANY (US) 1997-05-20 US disclosed
EP-0763011-A1 PROCESS FOR THE PREPARATION OF UNSATURATED AMINO COMPOUNDS Novartis AG (CH) 1997-03-19 EP disclosed
US-5502027-A ALGICIDES ROHM AND HAAS COMPANY (US) 1996-03-26 US disclosed
US-5238908-A HERBICIDAL GLUTARAMIC ACIDS AND DERIVATIVES ROHM AND HAAS COMPANY (US) 1993-08-24 US disclosed
US-5068365-A Herbicides TOSOH CORPORATION (JP) 1991-11-26 US disclosed
US-5053071-A For cereal crops E. I. DU PONT DE NEMOURS AND COMPANY (US) 1991-10-01 US disclosed
US-5017213-A Herbicides NIHON TOKUSHU NOYAKU SEIZO K. K. (JP) 1991-05-21 US disclosed
EP-0415641-A1 Substituted glutaramic acids and derivatives ROHM AND HAAS COMPANY (US) 1991-03-06 EP disclosed
US-4948418-A PREEMERGENCE AND POSTEMERGENCE HERBICIDES; WEED CONTROL, RICE, WHEAT, BARLEY, CORN, SOYBEANS, BEETS AND COTTON E. I. DU PONT DE NEMOURS AND COMPANY (US) 1990-08-14 US disclosed
EP-0351641-A1 1-Phenylpyrrole NIHON BAYER AGROCHEM K.K. (JP) 1990-01-24 EP disclosed
US-4881967-A Heterocyclic 2,3-dihydrobenzofuran herbicides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1989-11-21 US disclosed
EP-0326764-A2 Hexahydrophthalic anilide derivatives and herbicide compositions containing the same Tosoh Corporation (JP) 1989-08-09 EP disclosed
EP-0271170-A2 Herbicidal substituted benzofurans and benzopyrans SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1988-06-15 EP disclosed