SCHEMBL8359243

SCHEMBL8359243

O=C(CCN1CCc2ccccc2C1)N1CCc2[nH]c(=O)c3cc(F)ccc3c2C1

nearest known ligand 0.75

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 10/20 0.75
PRMT5 O14744 1/20 0.46
WDR77 Q9BQA1 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
BAZ2B Q9UIF8 1/20 0.45
HTR1A P08908 1/20 0.45
DRD2 P14416 1/20 0.45
HTR2A P28223 1/20 0.45
HTR7 P34969 1/20 0.45
HRH1 P35367 1/20 0.45
DRD3 P35462 1/20 0.45
HTR2B P41595 1/20 0.45
APAF1 O14727 1/20 0.44
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8362890 0.90 PARP1 (0.76) PARP1ALDH1A1
SCHEMBL8359236 0.86 PARP1 (1.00) PARP1BAZ2BALDH1A1GAA
SCHEMBL8359252 0.86 SIGMAR1 (0.56) PARP1HTR1ADRD2HTR2AHTR7
SCHEMBL14444052 0.82 PARP1 (0.76) PARP1CYP1A2CYP3A4CYP2C19BAZ2B
SCHEMBL8359419 0.81 PARP1 (0.74) PARP1BAZ2BALDH1A1GAA
SCHEMBL8359238 0.80 PARP1 (1.00) PARP1BAZ2BALDH1A1GAA
SCHEMBL8363079 0.80 PARP1 (0.74) PARP1ALDH1A1GAA
SCHEMBL8359241 0.79 PARP1 (0.71) PARP1CYP1A2CYP3A4CYP2C19BAZ2B
SCHEMBL8362899 0.78 PARP1 (0.84) PARP1BAZ2BALDH1A1GAA
SCHEMBL8359249 0.78 PARP1 (0.66) PARP1CYP1A2CYP3A4CYP2C19BAZ2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7247641-B2 Compounds, derivatives, compositions, preparation and uses MGI GP, INC. (US) 2007-07-24 US disclosed
US-7247641-B2 Compounds, derivatives, compositions, preparation and uses MGI GP, INC. (US) 2007-07-24 US disclosed
WO-2003014121-A9 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARM INC (US) 2004-03-25 WO disclosed
WO-2003014121-A1 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARMACEUTICALS INC. (US) 2003-02-20 WO disclosed