SCHEMBL8359448

SCHEMBL8359448

Cc1cc(N)c2cc(NC(=O)c3ccccc3)ccc2n1

nearest known ligand 0.86

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 6/20 0.73
MMP1 P03956 3/20 0.73
GNG2 P59768 2/20 0.73
GNB1 P62873 2/20 0.73
MEN1 O00255 1/20 0.73
ALOX15 P16050 1/20 0.73
BLM P54132 1/20 0.73
KMT2A Q03164 1/20 0.73
OPRL1 P41146 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5848272 0.94 MMP9 (0.71) MMP9MMP1GNG2GNB1MEN1
SCHEMBL3237985 0.90 MMP9 (0.68) MMP9MMP1GNG2GNB1MEN1
SCHEMBL5553600 0.90 MMP9 (0.70) MMP9MMP1GNG2GNB1MEN1
SCHEMBL8515694 0.89 MMP9 (0.68) MMP9MMP1GNG2GNB1MEN1
SCHEMBL3240190 0.87 MMP9 (0.65) MMP9MMP1GNG2GNB1MEN1
SCHEMBL5354568 0.86 MMP9 (0.68) MMP9MMP1GNG2GNB1MEN1
SCHEMBL3648167 0.85 NPC1 (0.67) MMP9MMP1GNG2GNB1MEN1
SCHEMBL8359605 0.85 GNG2 (0.83) MMP9MMP1GNG2GNB1MEN1
Aminoquinuride SCHEMBL29852258 0.85 GNG2 (1.00) MMP9MMP1GNG2GNB1MEN1
Aminoquinuride SCHEMBL321401 0.85 GNG2 (1.00) MMP9MMP1GNG2GNB1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998027815-A1 SUBSTITUTED AMINOQUINOLINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 1998-07-02 WO claimed
US-5919776-A ANTIINFLAMMATORY AGENT; AUTOIMMUNE DISEASE MERCK & CO., INC. (US) 1999-07-06 US disclosed
WO-1998027815-A1 SUBSTITUTED AMINOQUINOLINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 1998-07-02 WO disclosed