SCHEMBL8359595

SCHEMBL8359595

Cc1cc(OCCBr)cc2sc(-c3ccccn3)nc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.45
NPC1 O15118 4/20 0.45
RAB9A P51151 3/20 0.45
ALDH1A1 P00352 3/20 0.45
TP53 P04637 1/20 0.45
TSHR P16473 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HSD17B10 Q99714 1/20 0.45
LMNA P02545 2/20 0.40
MIF P14174 1/20 0.40
GABRA1 P14867 1/20 0.40
MAPT P10636 2/20 0.40
HTT P42858 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
KMT2A Q03164 2/20 0.39
F2RL3 Q96RI0 3/20 0.38
PDE10A Q9Y233 1/20 0.38
GAA P10253 1/20 0.38
ATM Q13315 1/20 0.37
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8359494 0.84 KDM4E (0.50) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL8552030 0.82 HTT (0.40) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL8356700 0.76 HTT (0.46) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL8358031 0.76 KDM4E (0.53) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL8050339 0.68 RAB9A (0.60) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL11782932 0.67 RAB9A (0.63) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL21474665 0.67 KDM4E (0.52) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL21474653 0.66 KDM4E (0.53) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL23954341 0.65 KDM4E (0.77) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL2958879 0.65 MIF (0.60) KDM4ENPC1RAB9AALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919807-A ANTICHOLESTEROL AGENTS DR. KARL THOMAE GMBH (DE) 1999-07-06 US disclosed
EP-0824529-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-02-25 EP disclosed
WO-1996035681-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-11-14 WO disclosed