SCHEMBL8362169

SCHEMBL8362169

NC(=O)N1CCN(c2ncccn2)CC1

nearest known ligand 0.65

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.58
ALDH1A1 P00352 5/20 0.55
L3MBTL1 Q9Y468 2/20 0.55
GAA P10253 1/20 0.55
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
SLC6A7 Q99884 3/20 0.54
TSHR P16473 1/20 0.54
HSD17B10 Q99714 1/20 0.54
PKM P14618 1/20 0.53
CYP2C19 P33261 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27580589 0.84 KDM4E (0.62) KDM4EALDH1A1L3MBTL1GAAMEN1
SCHEMBL27638766 0.83 HTR1A (0.42) KDM4EALDH1A1L3MBTL1GAAMEN1
SCHEMBL2856220 0.82 GAA (0.61) KDM4EALDH1A1L3MBTL1GAAMEN1
SCHEMBL9558198 0.81 MEN1 (0.59) KDM4EALDH1A1L3MBTL1GAAMEN1
SCHEMBL1919434 0.81 MEN1 (0.73) KDM4EALDH1A1L3MBTL1GAAMEN1
SCHEMBL5888121 0.80 HSD17B10 (0.56) KDM4EALDH1A1L3MBTL1GAAMEN1
SCHEMBL5888051 0.80 KDM4E (0.60) KDM4EALDH1A1L3MBTL1GAAMEN1
Triethylenemelamine SCHEMBL21332502 0.79 HTT (0.48) KDM4EALDH1A1L3MBTL1MEN1KMT2A
Hydrochloric Acid SCHEMBL29207063 0.79 KDM4E (0.49) KDM4EALDH1A1L3MBTL1GAAMEN1
SCHEMBL1270156 0.79 ALDH1A1 (0.66) KDM4EALDH1A1L3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119816492-A TRPV2 channel blocker and use thereof 伊契洛夫科技有限公司 2025-04-11 CN claimed
CN-119816492-A TRPV2 channel blocker and use thereof 伊契洛夫科技有限公司 2025-04-11 CN disclosed
EP-3564253-A1 ANTIDEPRESSANT COMPOUND AND PREPARATION METHOD AND APPLICATION THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2019-11-06 EP disclosed
EP-0810991-B1 1-ARYL-2-ACYLAMINO-ETHANE COMPOUNDS AND THEIR USE AS NEUROKININ ESPECIALLY NEUROKININ 1 ANTAGONISTS NOVARTIS AG (CH) 1999-04-14 EP disclosed
EP-0810991-A1 1-ARYL-2-ACYLAMINO-ETHANE COMPOUNDS AND THEIR USE AS NEUROKININ ESPECIALLY NEUROKININ 1 ANTAGONISTS Novartis AG (CH) 1997-12-10 EP disclosed
WO-1996026183-A1 1-ARYL-2-ACYLAMINO-ETHANE COMPOUNDS AND THEIR USE AS NEUROKININ ESPECIALLY NEUROKININ 1 ANTAGONISTS NOVARTIS AG (CH) 1996-08-29 WO disclosed