SCHEMBL8362256

SCHEMBL8362256

CC(C)(C)OC(=O)NC(CCC(=O)O)c1ccc2ccccc2c1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GABRB1 P18505 1/20 0.52
GABRB2 P47870 1/20 0.52
CTSB P07858 1/20 0.49
CTSS P25774 1/20 0.49
CTSK P43235 1/20 0.49
UTS2R Q9UKP6 13/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13802924 0.89 GABRB1 (0.53) GABRB1GABRB2CTSBCTSSCTSK
SCHEMBL9295219 0.89 GABRB1 (0.50) GABRB1GABRB2CTSBCTSSCTSK
SCHEMBL21715586 0.87 GABRB1 (0.48) GABRB1GABRB2CTSBCTSSCTSK
SCHEMBL5848532 0.86 GABRB1 (0.52) GABRB1GABRB2CTSBCTSSCTSK
SCHEMBL5676217 0.86 GABRB1 (0.52) GABRB1GABRB2CTSBCTSSCTSK
SCHEMBL4583120 0.86 CTSK (0.53) GABRB1GABRB2CTSBCTSSCTSK
SCHEMBL7299702 0.83 GABRB1 (0.49) GABRB1GABRB2CTSBCTSSCTSK
SCHEMBL4927517 0.81 JAK2 (0.46) GABRB1GABRB2CTSSCTSK
SCHEMBL4958137 0.81 CTSL (0.49) CTSSCTSK
SCHEMBL28389834 0.80 GABRB1 (0.54) GABRB1GABRB2CTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1081625-C 1 -aryl -2 -acylamino-ethane compounds and their use as neurokinin especially neurokinin 1 antagonists NOVARTIS AG (CH) 2002-03-27 CN disclosed
EP-0810991-B1 1-ARYL-2-ACYLAMINO-ETHANE COMPOUNDS AND THEIR USE AS NEUROKININ ESPECIALLY NEUROKININ 1 ANTAGONISTS NOVARTIS AG (CH) 1999-04-14 EP disclosed
CN-1175944-A 1 -aryl -2 -acylamino-ethane compounds and their use as neurokinin especially neurokinin 1 antagonists CIBA GEIGY AG (CH) 1998-03-11 CN disclosed