SCHEMBL8364174

SCHEMBL8364174

CC(=O)Oc1ccc2ncnc(Nc3ccc(OCc4ccccc4)cc3)c2c1

nearest known ligand 0.75

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 16/20 0.75
ERBB2 P04626 13/20 0.75
ERBB4 Q15303 2/20 0.67
AURKB Q96GD4 2/20 0.67
CHEK2 O96017 1/20 0.67
ROS1 P08922 1/20 0.67
FLT3 P36888 1/20 0.67
CLK4 Q9HAZ1 1/20 0.67
MKNK2 Q9HBH9 1/20 0.67
TTBK1 Q5TCY1 1/20 0.54
TTBK2 Q6IQ55 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8810261 0.99 EGFR (0.74) EGFRERBB2ERBB4AURKBCHEK2
Hydrochloric Acid SCHEMBL8811372 0.91 EGFR (0.65) EGFRERBB2ERBB4AURKBCHEK2
SCHEMBL5144877 0.89 EGFR (0.70) EGFRERBB2CLK4
SCHEMBL8809158 0.89 EGFR (0.67) EGFRERBB2ERBB4AURKBCHEK2
SCHEMBL8154615 0.88 EGFR (0.77) EGFRERBB2ERBB4AURKBCHEK2
SCHEMBL8807778 0.88 EGFR (0.77) EGFRERBB2ERBB4AURKBCHEK2
SCHEMBL1387244 0.86 EGFR (1.00) EGFRERBB2ERBB4AURKBCHEK2
Hydrochloric Acid SCHEMBL8808379 0.85 EGFR (0.98) EGFRERBB2ERBB4AURKBCHEK2
SCHEMBL8363497 0.85 EGFR (1.00) EGFRERBB2ERBB4AURKBCHEK2
SCHEMBL6663913 0.84 EGFR (0.79) EGFRERBB2ERBB4AURKBCHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999035132-A1 HETEROCYCLIC COMPOUNDS GLAXO GROUP LIMITED (GB) 1999-07-15 WO disclosed
EP-0782570-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1997-07-09 EP disclosed
WO-1996009294-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1996-03-28 WO disclosed