SCHEMBL8809158

SCHEMBL8809158

CC(=O)Oc1cc2ncnc(Nc3ccc(OCc4ccccc4)cc3)c2cc1OC(C)=O

nearest known ligand 0.67

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EGFR P00533 14/20 0.67
ERBB2 P04626 8/20 0.67
ERBB4 Q15303 3/20 0.67
AURKB Q96GD4 3/20 0.62
CHEK2 O96017 1/20 0.62
ROS1 P08922 1/20 0.62
FLT3 P36888 1/20 0.62
CLK4 Q9HAZ1 1/20 0.62
MKNK2 Q9HBH9 1/20 0.62
RIPK2 O43353 1/20 0.56
EPHB2 P29323 1/20 0.56
KDR P35968 2/20 0.56
AURKA O14965 1/20 0.54
RET P07949 1/20 0.54
PDGFRB P09619 1/20 0.54
TTBK1 Q5TCY1 1/20 0.53
TTBK2 Q6IQ55 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13404528 0.93 EGFR (0.71) EGFRERBB2ERBB4AURKBFLT3
SCHEMBL8364174 0.89 EGFR (0.75) EGFRERBB2ERBB4AURKBCHEK2
Hydrochloric Acid SCHEMBL8811372 0.88 EGFR (0.65) EGFRERBB2ERBB4AURKBCHEK2
Hydrochloric Acid SCHEMBL8810261 0.88 EGFR (0.74) EGFRERBB2ERBB4AURKBCHEK2
SCHEMBL17836949 0.87 EGFR (0.70) EGFRAURKBFLT3RIPK2EPHB2
SCHEMBL242224 0.86 EGFR (0.78) EGFRERBB2ERBB4AURKBCHEK2
SCHEMBL30141491 0.86 EGFR (0.78) EGFRERBB2ERBB4AURKBCHEK2
Hydrochloric Acid SCHEMBL8809813 0.85 EGFR (0.76) EGFRERBB2ERBB4AURKBCHEK2
Trifluoroacetic Acid SCHEMBL20494312 0.84 EGFR (0.72) EGFRERBB2ERBB4AURKBCHEK2
Hydrochloric Acid SCHEMBL8810888 0.84 EGFR (0.68) EGFRERBB2ERBB4AURKBCHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0782570-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1997-07-09 EP disclosed
WO-1996009294-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1996-03-28 WO disclosed